Front cover pg X001; DOI: 10.1039/P199500FX001 |
Contents pages pg P001; DOI: 10.1039/P199500FP001 |
(R)-(+)-3-Amino-2-phenylpropanoic acid: a revised absolute configuration based on an enantioselective synthesis and an X-ray crystal structure of the salt with (1S)-(+)-camphor-10-sulfonic acid Alice A. D'Souza Majid Motevalli Andrew J. Robinson and Peter B. Wyatt pg 1; DOI: 10.1039/P19950000001 |
Platinum-catalysed addition of trimethylgermane to 1-trimethylsilylalk-1-ynes: a convenient synthesis of functionalised 2-trimethylgermylalk-1-enes Edward Piers and René Lemieux pg 3; DOI: 10.1039/P19950000003 |
Back cover pg X003; DOI: 10.1039/P199500BX003 |
Nickel-catalysed substitutions of aryl tert-butyl sulfones with organometallic reagents: synthesis of ortho-substituted unsymmetrical biaryls Jonathan Clayden J. Jonathan A. Cooney and Marc Julia pg 7; DOI: 10.1039/P19950000007 |
Improved synthesis of isoguanosine and 6-substituted xanthosine derivatives Lorenzo De Napoli Daniela Montesarchio Gennaro Piccialli Ciro Santacroce and Michela Varra pg 15; DOI: 10.1039/P19950000015 |
Radical cyclisation in heterocycle synthesis. Part 1. Sulfanyl radical addition–cyclisation of dienylamides for lactam synthesis Takeaki Naito Yuko Honda Okiko Miyata and Ichiya Ninomiya pg 19; DOI: 10.1039/P19950000019 |
(Halogenomethyl)phenyl -D-glucopyranosides as enzyme-activated irreversible inhibitors of yeast -glucosidase and potential anti-HIV agents Josie C. Briggs Alan H. Haines and Richard J. K. Taylor pg 27; DOI: 10.1039/P19950000027 |
Additivity relationships in the carbon-13 nuclear magnetic resonance spectra of polyhydroxy steroids Masaru Kobayashi pg 33; DOI: 10.1039/P19950000033 |
[3 + 2] Cycloadditions of carbonyl oxides to imines: an alternative approach to the synthesis of 1,2,4-dioxazolidines Kevin J. McCullough Mitsuyuki Mori Toshihiko Tabuchi Hideyuki Yamakoshi Shigekazu Kusabayashi and Masatomo Nojima pg 41; DOI: 10.1039/P19950000041 |
Photoinduced molecular transformations. Part 152. Ring expansion based on a sensitized [2 + 2] photoaddition of enol ethers of cyclic ketones with olefins, followed by a -scission of alkoxyl radicals generated from the resulting cyclobutanols. Two-carbon ring expansion of -indanone, -tetralone and -suberone Hiroshi Suginome Toshihiro Takeda Masahito Itoh Yutaka Nakayama and Kazuhiro Kobayashi pg 49; DOI: 10.1039/P19950000049 |
Photoinduced molecular transformations. Part 153. Long-range intramolecular hydroxylation of C(25) of the cholestane side chain Kazuhiko Orito Shinji Sato and Hiroshi Suginome pg 63; DOI: 10.1039/P19950000063 |
Photoinduced molecular transformations. Part 155. General synthesis of macrocyclic ketones based on a ring expansion involving a selective -scission of alkoxyl radicals, its application to a new synthesis of ()-isocaryophyllene and ()-caryophyllene, and a conformational analysis of the two sesquiterpenes and the radical intermediate in the synthesis by MM3 calculations Hiroshi Suginome Takahiko Kondoh Camelia Gogonea Vishwakarma Singh Hitoshi Got and Eiji sawa pg 69; DOI: 10.1039/P19950000069 |
Design and synthesis of new bile acid-based macrocycles Uday Maitra and S. Balasubramanian pg 83; DOI: 10.1039/P19950000083 |
Instructions for authors (1995) pg vii; DOI: 10.1039/P19950000vii |
IUPAC publications on nomenclature and symbolism pg xxv; DOI: 10.1039/P19950000xxv |
Conference diary pg xxxi; DOI: 10.1039/P1995000xxxi |
Front cover pg X005; DOI: 10.1039/P199500FX005 |
Back cover pg X007; DOI: 10.1039/P199500BX007 |
Contents pages pg P009; DOI: 10.1039/P199500FP009 |
Back matter pg P017; DOI: 10.1039/P199500BP017 |
Lipase-catalysed Baeyer–Villiger reactions Stephanie C. Lemoult Paul F. Richardson and Stanley M. Roberts pg 89; DOI: 10.1039/P19950000089 |
A convenient and general synthesis of alkanediyl diphenols Cordula Grüttner Volker Böhmer Rosemarie Assmus and Sabine Scherf pg 93; DOI: 10.1039/P19950000093 |
Synthesis of acyl(phenylselanyl)methylidene(triphenyl)-5-arsanes and their Wittig-type reactions Zhi-Zhen Huang Xian Huang and Yao-Zeng Huang pg 95; DOI: 10.1039/P19950000095 |
Synthetic applications of arenetricarbonylchromium(0) complexes: the synthesis of polyfunctionalised thiophenes Michael S. Loft Timothy J. Mowlem and David A. Widdowson pg 97; DOI: 10.1039/P19950000097 |
Enhanced lability of -silyl groups in thiophenetricarbonylchromium(0) complexes Michael S. Loft Timothy J. Mowlem David A. Widdowson and David J. Williams pg 105; DOI: 10.1039/P19950000105 |
Asymmetric synthesis of (1R,1R)- and (1S,1S)-bis(1-arylethyl)amines by way of a diastereoselective addition to chiral imines and oxaxolidines with organometallic reagents Kimio Higashiyama Hiroaki Inoue Takayasu Yamauchi and Hiroshi Takahashi pg 111; DOI: 10.1039/P19950000111 |
Optical resolution and absolute stereochemistry of trans-2,5-dimethyl-1-phenyl-1-silacyclopentane Hai-Shan Dang Brian P. Roberts and Derek A. Tocher pg 117; DOI: 10.1039/P19950000117 |
Effect of molecular sieves on the formation and acid-catalysed mono- and bis-cyclization of N-arylimines: easy entry to polycyclic ring systems by a novel cascade reaction Oliver Temme and Sabine Laschat pg 125; DOI: 10.1039/P19950000125 |
5,9-Methanobenzoannulenamines. Part 1. Improved synthesis of 11-amino-5,9-methanobenzo[8]annulenes Iain M. Gilbert (the late) Colin L. Hewett Duncan R. Rae James Redpath (the late) David S. Savage and Thomas Sleigh pg 133; DOI: 10.1039/P19950000133 |
Stereocontrol in the nucleophilic epoxidation of -(1-hydroxyalkyl)-,-unsaturated sulfones Richard F. W. Jackson Stephen P. Standen William Clegg and Andrew McCamley pg 141; DOI: 10.1039/P19950000141 |
Control of diastereofacial selectivity in the nucleophilic epoxidation of -oxygenated ,-unsaturated sulfones Richard F. W. Jackson Stephen P. Standen and William Clegg pg 149; DOI: 10.1039/P19950000149 |
Stereospecific synthesis of -deuteriated -amino acids: regiospecific deuteriation of chiral 3-isopropyl-2,5-dimethoxy-3,6-dihydropyrazines Janet E. Rose Paul D. Leeson and David Gani pg 157; DOI: 10.1039/P19950000157 |
Carotenoids and related polyenes. Part 2. Photoisomerization of an allenic carotenoid, peridinin, and allenic model compounds Yumiko Yamano Sanae Sumiya and Masayoshi Ito pg 167; DOI: 10.1039/P19950000167 |
On the mechanism for the phototransformation of 3-alkoxy-2-(2-furyl)-4-oxo-4H-1-benzopyrans Satish C. Gupta Ashok Saini Devinder Kumar Narender S. Yadav Kuldeep Chand Satbir Mor and Som N. Dhawan pg 177; DOI: 10.1039/P19950000177 |
Corrigenda Brindaban C. Ranu Manika Saha Sanjay Bhar R. Rathore J. S. Kim and J. K. Kochi pg 183; DOI: 10.1039/P19950000183 |
Conference diary pg viia; DOI: 10.1039/P1995000viia |
Front cover pg X009; DOI: 10.1039/P199500FX009 |
Back cover pg X011; DOI: 10.1039/P199500BX011 |
Contents pages pg P019; DOI: 10.1039/P199500FP019 |
A superior procedure for generation of substituted benzyllithiums from the corresponding chlorides Keith Smith and Duanjie Hou pg 185; DOI: 10.1039/P19950000185 |
Facile synthesis of dihydrofurans by the cerium(IV) ammonium nitrate mediated oxidative addition of 1,3-dicarbonyl compounds to cyclic and acyclic alkenes. Relative superiority over the manganese(III) acetate mediated process Vijay Nair and Jessy Mathew pg 187; DOI: 10.1039/P19950000187 |
PbCl2/Ga bimetal redox system-mediated carbon–carbon bond formation reactions between carbonyl compounds and ethyl trichloroacetate and iodoacetonitrile Xiao-Lin Zhang Ying Han Wen-Tian Tao and Yao-Zeng Huang pg 189; DOI: 10.1039/P19950000189 |
Synthesis of alkyl and aryl substituted buta-1,2,3-trienes Hak-Fun Chow Xiao-Ping Cao and Man-Kit Leung pg 193; DOI: 10.1039/P19950000193 |
Studies of chromenes. Part 11. 3-Substitution of 7-methoxy-2,2-dimethylchroman-4-one without ring opening via 3-bromination Robert K. Akuamoah Philip E. Brown Wafa Y. Marcus and John E. Steele pg 197; DOI: 10.1039/P19950000197 |
Azoniaazulenes. Part 7. Functionalisation of 10H-azepino[1,2-a]indoles Gurnos Jones Michael W. Kempa Michael B. Hursthouse and K. Abdul Malik pg 203; DOI: 10.1039/P19950000203 |
Preparation and enantiomer recognition behaviour of azophenolic crown ethers containing cis-cyclohexane-1,2-diol as the chiral centre Koichiro Naemura Sachiko Takeuchi Keiji Hirose Yoshito Tobe Takahiro Kaneda and Yoshiteru Sakata pg 213; DOI: 10.1039/P19950000213 |
Excitatory amino acids. Synthesis of (RS)-2-amino-3-(5-cyclopropyl-3-hydroxyisoxazol-4-yl)propionic acid, a new potent and specific AMPA receptor agonist Niels Skjærbæk Bjarke Ebert Erik Falch Lotte Brehm and Povl Krogsgaard-Larsen pg 221; DOI: 10.1039/P19950000221 |
Short synthetic route to congeners of the undecose antibiotic herbicidin John R. Bearder Mark L. Dewis and Donald A. Whiting pg 227; DOI: 10.1039/P19950000227 |
Facile construction of the 1-phenylnaphthyl skeleton via an ester-mediated nucleophilic aromatic substitution reaction. Applications to the synthesis of phenylnaphthalide lignans Tetsutaro Hattori Hideyuki Tanaka Yoshikazu Okaishi and Sotaro Miyano pg 235; DOI: 10.1039/P19950000235 |
Preparation of N-hydroxyazoles by oxidation of azoles Mikael Begtrup and Per Vedsø pg 243; DOI: 10.1039/P19950000243 |
Antitumour imidazotetrazines. Part 31. The synthesis of isotopically labelled temozolomide and a multinuclear (1H, 13C, 15N) magnetic resonance investigation of temozolomide and mitozolomide Richard T. Wheelhouse Derry E. V. Wilman William Thomson and Malcolm F. G. Stevens pg 249; DOI: 10.1039/P19950000249 |
Reactions of tetrasulfur tetranitride with aryl dibromomethyl ketones: one-pot synthesis of 3-aroylformamido-4-aryl-1,2,5-thiadiazoles and their reactions Kyongtae Kim Jaeeock Cho and Sung Cheol Yoon pg 253; DOI: 10.1039/P19950000253 |
Regioselectivity in the reductive cleavage of pyrogallol derivatives: reductive electrophilic substitution of acetals of 2,3-dimethoxyphenol Ugo Azzena Giovanni Melloni and Luisa Pisano pg 261; DOI: 10.1039/P19950000261 |
Novel preparation of 3-alkyl-5-hydroxy-5-per(poly)fluoroalkyl-4,5-dihydroisoxazoles Jian Chen and Chang-Ming Hu pg 267; DOI: 10.1039/P19950000267 |
Stereoselective radical additions of -oxy-,-unsaturated ester derivatives; 1,2-asymmetric induction in acyclic and cyclisation systems Tsutomu Morikawa Yoshiaki Washio Susumu Harada Ryo Hanai Takashi Kayashita Hisako Nemoto Motoo Shiro and Takeo Taguchi pg 271; DOI: 10.1039/P19950000271 |
Conference diary pg viib; DOI: 10.1039/P1995000viib |
Front cover pg X013; DOI: 10.1039/P199500FX013 |
Back cover pg X015; DOI: 10.1039/P199500BX015 |
Contents pages pg P027; DOI: 10.1039/P199500FP027 |
Back matter pg P039; DOI: 10.1039/P199500BP039 |
Proof that acetic acid is extruded during biosynthesis of vitamin B12 in Pseudomonas denitrificans Yongfu Li N. Patrick J. Stamford and Alan R. Battersby pg 283; DOI: 10.1039/P19950000283 |
Diastereocontrol in the reaction of amide-homoenolates with aromatic aldehydes Satoshi Sakami Takashi Houkawa Morio Asaoka and Hisashi Takei pg 285; DOI: 10.1039/P19950000285 |
Synthesis of 11C-labelled ketones via carbonylative coupling reactions using [11C]carbon monoxide Yvonne Andersson and Bengt Långström pg 287; DOI: 10.1039/P19950000287 |
Nitration of nonactivated arenes with a ternary system NO–NO2–O2. Mechanistic implications of the Kyodai-nitration Hitomi Suzuki and Tadashi Mori pg 291; DOI: 10.1039/P19950000291 |
Porphyrin–phenothiazine hybrid molecules: marked dependence of light induced nuclease activity on the linker moiety Goverdhan Mehta Thota Sambaiah Bhaskar G. Maiya Mallena Sirish and Aparna Dattagupta pg 295; DOI: 10.1039/P19950000295 |
Synthesis and anti-HIV-1 activity of bis-ketol AZT monophosphates Gerald F. Koser Yali Huang Kuanchiang Chen and Kim C. Calvo pg 299; DOI: 10.1039/P19950000299 |
Diastereoselectivity in the preparation of -silyl esters from -unsaturated esters and amides attached to chiral auxiliaries Ian Fleming and Nicholas D. Kindon pg 303; DOI: 10.1039/P19950000303 |
The phenyldimethylsilyl group as a masked hydroxy group Ian Fleming Rolf Henning David C. Parker Howard E. Plaut and Philip E. J. Sanderson pg 317; DOI: 10.1039/P19950000317 |
Ozone-mediated reaction of anilides and phenyl esters with nitrogen dioxide: enhanced ortho-reactivity and mechanistic implications Hitomi Suzuki Atsuo Tatsumi Taro Ishibashi and Tadashi Mori pg 339; DOI: 10.1039/P19950000339 |
Some enantioselective borane reductions of prochiral ketones catalysed by polymer-supported oxazaborolidines bound via the boron atom Claude Caze Noureddine El Moualij Philip Hodge Christopher J. Lock and Jianbiao Ma pg 345; DOI: 10.1039/P19950000345 |
Development of a synthesis of lankacidins: stereoselective synthesis of the -lactone fragment Eric J. Thomas and Andrew C. Williams pg 351; DOI: 10.1039/P19950000351 |
Development of a synthesis of lankacidins: synthesis of the C(14)–C(6) fragment and introduction of the C(10)–C(13) diene Jane M. Roe and Eric J. Thomas pg 359; DOI: 10.1039/P19950000359 |
Synthesis of 7-benzylideneoctahydro-2H-pyrido[1,2-a]pyrazines, bicyclic analogues of the calcium antagonist flunarizine M. Ashty Saleh Frans Compernolle Suzanne Toppet and Georges J. Hoornaert pg 369; DOI: 10.1039/P19950000369 |
Photochemical isomerization of O-allyl and O-but-3-enyl thiocarbamates Masami Sakamoto Mitsuru Yoshiaki Masaki Takahashi Tsutomu Fujita and Shoji Watanabe pg 373; DOI: 10.1039/P19950000373 |
Hydroxyl-directed reduction of -hydroxycycloalkanones as a stereoselective route to 1,3-diols: X-ray crystal structure and structural features of (1R*,2R*,6S*)-2-[hydroxy(phenyl)methyl]cyclopentanol Stephen H. J. Thompson Mary F. Mahon Kieran C. Molloy Michael S. Hadley and Timothy Gallagher pg 379; DOI: 10.1039/P19950000379 |
Synthesis of a derivative of triangulene; the first non-kekul polynuclear aromatic Graeme Allinson Richard J. Bushby Jean-Louis Paillaud and Mark Thornton-Pett pg 385; DOI: 10.1039/P19950000385 |
Structure and relative stereochemistry of a new polycyclic alkaloid, asparagamine A, showing anti-oxytocin activity, isolated from Asparagus racemosus Toshikazu Sekine Fumio Ikegami Nobuaki Fukasawa Yumi Kashiwagi Tatsuo Aizawa Yuichi Fujii Nijsiri Ruangrungsi and Isamu Murakoshi pg 391; DOI: 10.1039/P19950000391 |
Synthesis of uridine derivatives containing strategically placed radical traps as potential inhibitors of ribonucleotide reductase Sandra P. Auguste and Douglas W. Young pg 395; DOI: 10.1039/P19950000395 |
Dithiasuccinoyl (Dts) amino-protecting group used in syntheses of 1,2-trans-amino sugar glycosides Ernst Meinjohanns Morten Meldal Hans Paulsen and Klaus Bock pg 405; DOI: 10.1039/P19950000405 |
Synthetic reactions of 2-(2-amino-3-cyano-4H-[1]benzopyran-4-yl)propane-1,3-dinitrile with reactive methylene compounds Conor N. O'Callaghan T. Brian H. McMurry and John E. O'Brien pg 417; DOI: 10.1039/P19950000417 |
Use of bis[2-(trialkylsilyl)ethyl]N,N-dialkylphosphoramidites for the synthesis of phosphate monoesters Kenneth C. Ross Daniel L. Rathbone William Thomson and Sally Freeman pg 421; DOI: 10.1039/P19950000421 |
Asymmetric reduction of prochiral aromatic ketones by borane–amine complexes in the presence of chiral amine–BF3 catalysts Mariappan Periasamy J. V. Bhaskar Kanth and Ch. Kishan Reddy pg 427; DOI: 10.1039/P19950000427 |
Rearrangement of S-methylbenzylsulfonium S-alkylides in non-basic media Tohru Tanzawa Miyuki Ichioka Naohiro Shirai and Yoshiro Sato pg 431; DOI: 10.1039/P19950000431 |
Modification of cyclodextrins by insertion of a heterogeneous sugar unit into their skeletons. Synthesis of 2-amino-2-deoxy--cyclodextrin from -cyclodextrin Nobuo Sakairi Lai-Xi Wang and Hiroyoshi Kuzuhara pg 437; DOI: 10.1039/P19950000437 |
Quinolinone cycloaddition as a potential synthetic route to dimeric quinoline alkaloids Stephen A. Barr Charles F. Neville (the late) Michael F. Grundon Derek R. Boyd John F. Malone and Timothy A. Evans pg 445; DOI: 10.1039/P19950000445 |
Selective electrophilic additions of mixed bifunctionalized trimethylenemethane dianion synthons George Majetich Hisaya Nishidie and Yong Zhang pg 453; DOI: 10.1039/P19950000453 |
Photochemical reactions of o-alkenylphenols and 1-alkenyl-2-naphthol with alkylamines: amination via photoinduced proton transfer Masahide Yasuda Tatsuya Sone Kimiko Tanabe and Kensuke Shima pg 459; DOI: 10.1039/P19950000459 |
Synthesis of perhydro-1,4-ethano-1,5-naphthyridine and perhydro-4,7-ethanopyrrolo[3,2-b]pyridine derivatives: potential NK1-receptor antagonists. X-Ray molecular structures of (4aR,8S,8aR)-6-oxo-8-phenylperhydro-1,4-ethano-1,5-naphthyridine and (4aR,7R,8R,8aR)-7,8-diphenylperhydro-1,4-ethano-1,5-naphthyridine Yevgeny Besidsky Kristina Luthman Alf Claesson Christopher J. Fowler Ingeborg Csöregh and Uli Hacksell pg 465; DOI: 10.1039/P19950000465 |
Synthesis and reactivity of 6-carbamoyl-5-phenyl-2,3,5,6-tetrahydro-1H-1,4-ethanobenzo[f]quinoline. X-Ray molecular structure of (4aR,5S,6R,10bR)-5-phenyl-2,3,4a,5,6,10b-hexahydro-1H-1,4-ethanobenzo[f]quinolin-6-yl acetate Yevgeny Besidsky Kristina Luthman Alf Claesson Ingeborg Csöregh and Uli Hacksell pg 475; DOI: 10.1039/P19950000475 |
The biosynthesis of hyoscyamine: the process by which littorine rearranges to hyoscyamine Richard J. Robins Nicola C. J. E. Chesters David O'Hagan Adrian J. Parr Nicholas J. Walton and Jack G. Woolley pg 481; DOI: 10.1039/P19950000481 |
The biosynthesis of tropic acid. Part 6. Enantioselective, intact incorporation of (R)-(+)-3-phenyllactic acid into the tropic acid ester alkaloids of Datura Morteza Ansarin and Jack G. Woolley pg 487; DOI: 10.1039/P19950000487 |
Acylation of aldo 1-pyrroline 1-oxides (4,5-dihydro-3H-pyrrole 1-oxides) and the oxidation of the resulting 3-acyloxy-1-pyrrolines (3-acyloxy-4,5-dihydro-3H-pyrroles) Neil J. Gibson and Alexander R. Forrester pg 491; DOI: 10.1039/P19950000491 |
Preparation and the acid- and base-catalysed isomerisation of 5,5-dimethyl-3-phenyl-1-pyrroline 1-oxide (5,5-dimethyl-3-phenyl-4,5-dihydro-3H-pyrrole 1-oxide): unprecedented acid-catalysed 1,3-oxygen migration Neil J. Gibson and Alexander R. Forrester pg 501; DOI: 10.1039/P19950000501 |
Preparation and benzoylation of 3-hydroxy-2,3,5,5-tetramethyl-1-pyrroline 1-oxide (3-hydroxy-2,3,5,5-tetramethyl-4,5-dihydro-3H-pyrrole 1-oxide) Neil J. Gibson Alexander R. Forrester and Charles Brown pg 507; DOI: 10.1039/P19950000507 |
Reaction of noracronycine and 1-hydroxy-3-methoxy-10-methylacridone with alkyl- and aryl-lithiums: formation of quinone methides Catherine Jolivet Christian Rivalle and Emile Bisagni pg 511; DOI: 10.1039/P19950000511 |
Conference diary pg xi; DOI: 10.1039/P199500000xi |
Front cover pg X017; DOI: 10.1039/P199500FX017 |
Back cover pg X019; DOI: 10.1039/P199500BX019 |
Contents pages pg P041; DOI: 10.1039/P199500FP041 |
Back matter pg P049; DOI: 10.1039/P199500BP049 |
Synthesis of C-glycofuranosides by the stereoselective reduction of hemiacetals Eguzkiñe Calzada Catherine A. Clarke Christine Roussin-Bouchard and Richard H. Wightman pg 517; DOI: 10.1039/P19950000517 |
One-pot syntheses of 3-cyanoindoles from 3-acyl- and 3-ethoxycarbonyl-1,2-dihydrocinnoline-1,2-dicarboximides Satoko Tanaka Kazuyoshi Seguchi and Akira Sera pg 519; DOI: 10.1039/P19950000519 |
Synthesis of substructures of soraphen A: formation of the enolate of benzyl propionate Bernard Loubinoux Jean-Luc Sinnes and Anthony C. O'Sullivan pg 521; DOI: 10.1039/P19950000521 |
Mechanistic studies of the palladium(II)–copper(II)-mediated demercuriation of cycloalkyl and cycloalkylmethyl systems Adam P. Wells and William Kitching pg 527; DOI: 10.1039/P19950000527 |
Synthesis and characterization of isomeric ,-bithienyls with -methylsulfanyl substituents Ugo Folli Dario Iarossi Mauro Montorsi Adele Mucci and Luisa Schenetti pg 537; DOI: 10.1039/P19950000537 |
The synthesis of precisely structured polyurethanes. Part 1. Monomer synthesis Alistair A. Denholm Maurice H. George Helen C. Hailes Peter J. Tiffin and David A. Widdowson pg 541; DOI: 10.1039/P19950000541 |
Selective alkylation and allylation of allylic halides by tetraorganoindates: regio- and stereo-selective synthesis of rosefuran and sesquirosefuran Shuki Araki Shun-Ji Jin and Yasuo Butsugan pg 549; DOI: 10.1039/P19950000549 |
Chemo–enzymic synthesis of optically active ,-disubstituted -amino acids Weiguo Liu Paul Ray and Steven A. Benezra pg 553; DOI: 10.1039/P19950000553 |
Photoreactions of 1,3-dihydroisobenzofuran-1-thiones and 1,3-dihydro-2-benzothiophene-1-thiones with alkenes Takehiko Nishio pg 561; DOI: 10.1039/P19950000561 |
Synthesis of 4-hydroxy-15-oxaandrost-4-en-3-one and other potential aromatase inhibitors from sandaracopimaric acid M. Bordell Martín A. Fernández Mateos and R. Rubio González pg 569; DOI: 10.1039/P19950000569 |
Synthesis of water-soluble sugar derivatives of combretastatin A-4 Richard T. Brown Brian W. Fox John A. Hadfield Alan T. McGown Stephen P. Mayalarp George R. Pettit and Julie A. Woods pg 577; DOI: 10.1039/P19950000577 |
Constituents of Nothapodytes foetida Angela Pirillo Luisella Verotta Pierluigi Gariboldi Elisabetta Torregiani and Ezio Bombardelli pg 583; DOI: 10.1039/P19950000583 |
Synthesis and Diels–Alder reactions of thioisobenzofurans Jonathan H. Bailey Carolyn V. Coulter Andrew J. Pratt and Ward T. Robinson pg 589; DOI: 10.1039/P19950000589 |
Structure of conocephalenol, a sesquiterpenoid alcohol from the European liverwort Conocephalum conicum: determination of the absolute configuration by total synthesis Motoo Tori Katsuyuki Nakashima Yoshinori Asakawa Joseph D. Connolly Leslie J. Harrison David S. Rycroft Jagdemba Singh and Neill Woods pg 593; DOI: 10.1039/P19950000593 |
Palladium complex-catalysed carbocyclization–distannylation, –disilylation and –silastannylation of bis-dienes using distannanes, disilanes and silylstannanes Yasushi Obora Yasushi Tsuji Takeshi Kakehi Mitsunari Kobayashi Yoshihisa Shinkai Masahiro Ebihara and Takashi Kawamura pg 599; DOI: 10.1039/P19950000599 |
Conference diary pg viic; DOI: 10.1039/P1995000viic |
Front cover pg X021; DOI: 10.1039/P199500FX021 |
Back cover pg X023; DOI: 10.1039/P199500BX023 |
Contents pages pg P053; DOI: 10.1039/P199500FP053 |
SRN1 Synthesis of vic-dinitro compounds containing a nitrodioxane subunit René Beugelmans Ali Amrollah Madjdabadi Tawfik Gharbaoui and (the late) André Lechevallier pg 609; DOI: 10.1039/P19950000609 |
Synthesis and thermal reactivity of 2-azido-5-trimethylsilylthiophene and 2-azido-5-methylthiophene. The para-like substituent effect on fragmentation of the azido group Darren Davies Piero Spagnolo and Paolo Zanirato pg 613; DOI: 10.1039/P19950000613 |
Rearrangement and cyclo--elimination of N-substituted amidines using (diacetoxyiodo)benzene Christopher A. Ramsden and Helen L. Rose pg 615; DOI: 10.1039/P19950000615 |
A new catalytic transformation of diazo esters: hydride abstraction in dirhodium(II)-catalysed reactions Michael P. Doyle Alexey B. Dyatkin and Christopher L. Autry pg 619; DOI: 10.1039/P19950000619 |
Tetrathiafulvalene: a catalyst for sequential radical–polar reactions Rodney J. Fletcher Christopher Lampard John A. Murphy and Norman Lewis pg 623; DOI: 10.1039/P19950000623 |
Low-temperature addition of hydrogen polysulfides to olefins: formation of 2,2-dialkyl polysulfides from alk-1-enes and cyclic (poly)sulfides and polymeric organic sulfur compounds from ,-dienes Wim de Graaf Jaap S. Sinninghe Damsté and Jan W. de Leeuw pg 635; DOI: 10.1039/P19950000635 |
Synthesis of the selective muscarinic agonist (3R)-3-(6-chloropyrazin-2-yl)-1-azabicyclo [2.2.2] octane Michael S. Ashwood Andrew W. Gibson Peter G. Houghton Guy R. Humphrey D. Craig Roberts and Stanley H. B. Wright pg 641; DOI: 10.1039/P19950000641 |
Pigments of fungi. Part 40. Dermocanarins 1–3, unique naphthol- and naphthoquinone-anthraquinone dimers that contain a macrocyclic lactone ring from the fungus Dermocybe canaria Horak Melvyn Gill and Alberto Giménez pg 645; DOI: 10.1039/P19950000645 |
Preparation of 2-chlorobuta-1,3-dienes by dichlorocyclopropanation of allylsilanes followed by desilylation Michiharu Mitani Yosinori Kobayashi and Kikuhiko Koyama pg 653; DOI: 10.1039/P19950000653 |
Radio-iodinated gibberellin photoaffinity probes Michael H. Beale Richard Hooley Mervyn J. Lewis Sally J. Smith and Jane L. Ward pg 657; DOI: 10.1039/P19950000657 |
Reaction of 4a-methyl-2,3,4,4a-tetrahydro-1H-carbazole with Grignard reagents J. Gonzalo Rodríguez and Anahí Urrutia pg 665; DOI: 10.1039/P19950000665 |
Synthesis of [1,2,3-2,3-bis(benzyloxymethyl)cyclobutyl]imidazol-5-amines: important precursors to cyclobut-A derivatives Brian L. Booth and Paul R. Eastwood pg 669; DOI: 10.1039/P19950000669 |
Two synthetic routes to 2,3-dideoxy-3-C-(hydroxymethyl)-4-thionucleosides John Mann Allen J. Tench Alexander C. Weymouth-Wilson Sue Shaw-Ponter and Robert J. Young pg 677; DOI: 10.1039/P19950000677 |
Absolute stereochemistry of chinesin I and II Yoshinori Aramaki Kazuhiro Chiba and Masahiro Tada pg 683; DOI: 10.1039/P19950000683 |
Samarium(II) diiodide-mediated intermolecular aldol type reactions of phenacyl bromides with carbonyl compounds Yutaka Aoyagi Mizue Yoshimura Masako Tsuda Tomomasa Tsuchibuchi Saori Kawamata Hiroyuki Tateno Kazushi Asano Hiroko Nakamura Masako Obokata Akihiro Ohta and Yoshio Kodama pg 689; DOI: 10.1039/P19950000689 |
Synthesis of optically active azetidine-2,4-dicarboxylic acid and related chiral auxiliaries for asymmetric synthesis Jun'ichi Hoshino Junko Hiraoka Yasuo Hata Seiji Sawada and Yukio Yamamoto pg 693; DOI: 10.1039/P19950000693 |
Oxidation of imines to oxaziridines catalysed by transition metal complexes using molecular oxygen as the terminal oxidant Lars Martiny and Karl Anker Jørgensen pg 699; DOI: 10.1039/P19950000699 |
Synthesis and characterization of models for the bilin catabolites of chlorophylls using metallo--oxochlorins and -benzo[at]chlorins: comparison of macrocycle cleavage versus meso-oxochlorin formation Meden Isaac Mathias O. Senge and Kevin M. Smith pg 705; DOI: 10.1039/P19950000705 |
Preparation and oxidative doping studies of dithienyl polyenes stabilized by alkyl group substitution Charles W. Spangler and Mingqian He pg 715; DOI: 10.1039/P19950000715 |
Benzoannelated centropolyquinanes. Part 21. Centrohexaindane: three complementary syntheses of the highest member of the centropolyindane family Dietmar Kuck Andreas Schuster Bernd Paisdor and Detlef Gestmann pg 721; DOI: 10.1039/P19950000721 |
Conference diary pg viid; DOI: 10.1039/P1995000viid |
Front cover pg X025; DOI: 10.1039/P199500FX025 |
Back cover pg X027; DOI: 10.1039/P199500BX027 |
Contents pages pg P061; DOI: 10.1039/P199500FP061 |
Back matter pg P071; DOI: 10.1039/P199500BP071 |
A new method for the synthesis of N-phenyl-uracil and -pyrimidine nucleosides Tokumi Maruyama Keiichi Fujiwara and Mitsutoshi Fukuhara pg 733; DOI: 10.1039/P19950000733 |
Highly selective asymmetric hydrolysis of 2,2-disubstituted epoxides using lyophilized cells of Rhodococcus sp. NCIMB 11216 Ute Wandel Martin Mischitz Wolfgang Kroutil and Kurt Faber pg 735; DOI: 10.1039/P19950000735 |
Generation and reactions of butadienylthionium ions from 2-vinylcyclopropyl sulfoxides under Pummerer conditions Tadashi Kataoka Harutoshi Matsumoto Tetsuo Iwama Taizo Ito and Hiroshi Shimizu pg 737; DOI: 10.1039/P19950000737 |
A new and convenient one-pot synthesis of ,-unsaturated trifluoromethyl ketones Wei Sheng Huang and Cheng Ye Yuan pg 741; DOI: 10.1039/P19950000741 |
Synthesis and decomplexation of (-arene)(-cyclopentadienyl)-iron(II) hexafluorophosphates using microwave dielectric heating Qumars Dabirmanesh Sharon I. S. Fernando and Roger M. G. Roberts pg 743; DOI: 10.1039/P19950000743 |
A ketal Claisen rearrangement for -ketol isoprene unit elongation: application to a practical synthesis of sarcophytol A intermediate Hisao Takayanagi Shigeo Sugiyama and Yasuhiro Morinaka pg 751; DOI: 10.1039/P19950000751 |
A total synthesis of an antibacterial clerodane, 16-hydroxycleroda-3,13(14)Z-dien-15,16-olide Hisahiro Hagiwara Kazuhiro Inome and Hisashi Uda pg 757; DOI: 10.1039/P19950000757 |
Structure of cereulide, a cyclic dodecadepsipeptide toxin from Bacillus cereus and studies on NMR characteristics of its alkali metal complexes including a conformational structure of the K+ complex Sathorn Suwan Minoru Isobe Ikuko Ohtani Norio Agata Masashi Mori and Michio Ohta pg 765; DOI: 10.1039/P19950000765 |
Total synthesis of (+)-compactin by a double Michael protocol Hisahiro Hagiwara Takashi Nakano Masakazu Kon-no and Hisashi Uda pg 777; DOI: 10.1039/P19950000777 |
Development of a synthesis of lankacidins: an investigation into 17-membered ring formation Ernesto G. Mata and Eric J. Thomas pg 785; DOI: 10.1039/P19950000785 |
Adenine isosteres with bridgehead nitrogen. Part 1. Two independent syntheses of the [1,2,4]triazolo[1,5-a][1,3,5]triazine ring system leading to a range of substituents in the 2, 5 and 7 positions Peter W. R. Caulkett Geraint Jones Mary McPartlin Nigel D. Renshaw Sarah K. Stewart and Brian Wright pg 801; DOI: 10.1039/P19950000801 |
Mild thermal route to phthalimidonitrene and its reaction with activated benzenes to give 2H- and 3H-azepines; X-ray crystal structure analysis of an isolable 2H-azepine David W. Jones and Mark Thornton-Pett pg 809; DOI: 10.1039/P19950000809 |
An enantiospecific total synthesis of (+)-muricatacin Peter Somfai pg 817; DOI: 10.1039/P19950000817 |
Synthesis and stereochemistry of optically active telluronium ylides Nobumasa Kamigata Ayumi Matsuhisa Hideo Taka and Toshio Shimizu pg 821; DOI: 10.1039/P19950000821 |
Selective ether cleavages: simple routes yielding di- and tri-functional hexaalkoxytriphenylenes Fritz Closs Lukas Häußling Philippe Henderson Helmut Ringsdorf and Peter Schuhmacher pg 829; DOI: 10.1039/P19950000829 |
Synthesis based on cyclohexadienes. Part 17. Total synthesis of the sesquiterpenes of Eremophila georgei diels Natesan Selvakumar Seenivasaga N. Janaki Kakumanu Pramod and G. S. R. Subba Rao pg 839; DOI: 10.1039/P19950000839 |
Homochiral 2,3-epoxy sulfides—powerful new synthetic building blocks providing stereoselective access to 2,3-epoxy sulfoxides, 2,3-dihydroxy sulfoxides and (E)--hydroxy-,-unsaturated sulfoxides and sulfones. X-Ray molecular structure of rac-(2R*,3R*)-1-[(S*)-phenylsulfinyl] hexane-2,3-diol Andrew D. Westwell Mark Thornton-Pett and Christopher M. Rayner pg 847; DOI: 10.1039/P19950000847 |
Synthesis of bridged thiazolium salts as models for thiamin Finian J. Leeper and David H. C. Smith pg 861; DOI: 10.1039/P19950000861 |
Changes of enantioselectivity with the substrate ratio for the addition of diethylzinc to aldehydes using a catalyst coupled to a soluble polymer Claus Dreisbach Gisela Wischnewski Udo Kragl and Christian Wandrey pg 875; DOI: 10.1039/P19950000875 |
Free-radical cyclisations of 2-aminoalka-2,5-dienenitriles Chau-Chen Yang and Jim-Min Fang pg 879; DOI: 10.1039/P19950000879 |
Stereocontrolled synthesis of fluorosqualenes and fluoroepoxy-squalenes as inhibitors of squalene epoxidase and 2,3-oxidosqualene cyclase Maurizio Ceruti Simona Amisano Paola Milla Franca Viola Flavio Rocco Michel Jung and Luigi Cattel pg 889; DOI: 10.1039/P19950000889 |
Helically chiral thia- and diselena-quinquephenylophanes Karri Airola Stefan Bartram and Kari Rissanen pg 895; DOI: 10.1039/P19950000895 |
Syntheses of 2-ethyl-8-methyl-1,7-dioxaspiro[5.5]undecanols Mark F. Jacobs Bill D. Suthers Achim Hübener and William Kitching pg 901; DOI: 10.1039/P19950000901 |
Simple transphosphatidylation of phospholipids catalysed by a lipid-coated phospholipase D in organic solvents Yoshio Okahata Ken-ichi Niikura and Kuniharu Ijiro pg 919; DOI: 10.1039/P19950000919 |
Radical cyclisation route to furanolignans: short and stereoselective synthesis of ()-dihydrosesamin and ()-lariciresinol Gourhari Maiti Sankar Adhikari and Subhas Chandra Roy pg 927; DOI: 10.1039/P19950000927 |
Synthesis of 4,5,8-trimethoxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acid, an analogue of rhein with improved systemic exposure in the guinea pig W. Martin Owton Michael Brunavs Martin V. Miles David R. Dobson and David J. Steggles pg 931; DOI: 10.1039/P19950000931 |
Synthetic study of the highly potent and selective anti-platelet activating factor thiazolidin-4-one agents and related compounds Yoo Tanabe Hitomi Yamamoto Masanari Murakami Kazunori Yanagi Yoshino Kubota Hitomi Okumura Yuzuru Sanemitsu and Gohfu Suzukamo pg 935; DOI: 10.1039/P19950000935 |
Total synthesis of pterocarpan: ()-neorautenane Ricardo A. Lichtenfels Antonio L. Coelho and Paulo R. R. Costa pg 949; DOI: 10.1039/P19950000949 |
Synthesis of phenylalanine-based cyclic acylated enamino ester dipeptide analogues: inhibitors of -chymotrypsin. X-Ray molecular structure of (2S,4R)-4-benzyl-3-benzyloxycarbonyl-5-oxo-2-phenyloxazolidin-4-ylacetic acid Andrew D. Abell Mark D. Oldham and Jane M. Taylor pg 953; DOI: 10.1039/P19950000953 |
Conference diary pg ix; DOI: 10.1039/P199500000ix |
Front cover pg X029; DOI: 10.1039/P199500FX029 |
Back cover pg X031; DOI: 10.1039/P199500BX031 |
Contents pages pg P081; DOI: 10.1039/P199500FP081 |
Back matter pg P089; DOI: 10.1039/P199500BP089 |
Total synthesis of cis-clerodane diterpenoids: (–)-agelasine A and (+)-(3R,4S,5R,8S,9R,10S)-3,4-epoxyclerod-13-en-15,16-olide Edward Piers M. Livain Breau Yongxin Han Guy L. Plourde and Wen-Lung Yeh pg 963; DOI: 10.1039/P19950000963 |
Enzymes in organic synthesis: oxidoreductions Jim-Min Fang Chun-Hung Lin Curt W. Bradshaw and Chi-Huey Wong pg 967; DOI: 10.1039/P19950000967 |
Nucleophilic addition of lithio derivatives to 1-substituted benzo[c][2,7]naphthyridines (2,9-diazaphenanthrenes) Corinne Cochennec Patrick Rocca Francis Marsais Alain Godard and Guy Quéguiner pg 979; DOI: 10.1039/P19950000979 |
Synthesis of 6,7- and 6,7-aziridinoandrost-4-ene-3,17-diones and related compounds: potential aromatase inhibitors Vincent C. O. Njar Rolf W. Hartmann and Cecil H. Robinson pg 985; DOI: 10.1039/P19950000985 |
Novel synthesis of trifluoromethylated allylic phosphonates Yanchang Shen and Ming Qi pg 993; DOI: 10.1039/P19950000993 |
Synthesis of perfluoroalkylated heterocyclic phosphonates Yanchang Shen Jianhua Zheng Yuankang Xin Yugang Lin and Ming Qi pg 997; DOI: 10.1039/P19950000997 |
On the reactions of (vinylimino)phosphoranes and related compounds. Part 30. Short new synthesis of 5-azaazulene derivatives. Some comments on reactivities of (vinylimino)phosphoranes Makoto Nitta Yukio Iino Satoshi Mori and Tohru Takayasu pg 1001; DOI: 10.1039/P19950001001 |
1,2-Asymmetric induction in conjugate additions to nitroalkenes Anthony G. M. Barrett and David J. Rys pg 1009; DOI: 10.1039/P19950001009 |
Synthetic approaches to the angucycline antibiotics: the total syntheses of ()-rubiginone B1 and B2, ()-emycin A, and related analogues David S. Larsen and Michael D. O'Shea pg 1019; DOI: 10.1039/P19950001019 |
Regiospecific electrophilic substitution of aminoquinazolinones: directed lithiation of 3-(pivaloylamino)- and 3-(acetylamino)-2-methylquinazolin-4(3H)-ones Keith Smith Gamal A. El-Hiti Mohamed A. Abdo and Mohamed F. Abdel-Megeed pg 1029; DOI: 10.1039/P19950001029 |
A useful method for configurational assignment of vinyl sulfides; stereochemical reassessment of the radical addition of benzenethiol to alkynes Luisa Benati Laura Capella Pier Carlo Montevecchi and Piero Spagnolo pg 1035; DOI: 10.1039/P19950001035 |
Convenient and versatile synthesis of 3-(polyfluoroalkyl)pyrazoles Xiao-Qing Tang and Chang-Ming Hu pg 1039; DOI: 10.1039/P19950001039 |
Potential mechanism-based tyrosine kinase inhibitors. Part 1. Phosphorylation chemistry of pyridine N-oxides David M. Andrews Timothy C. M. Page Josephine M. Peach and Andrew J. Pratt pg 1045; DOI: 10.1039/P19950001045 |
Oligomeric isoflavonoids. Part 3. Daljanelins A–D, the first pterocarpan- and isoflavanoid-neoflavonoid analogues J. Albert Ferreira Janetta W. Nel E. Vincent Brandt Barend C. B. Bezuidenhoudt and Daneel Ferreira pg 1049; DOI: 10.1039/P19950001049 |
Catalytic oxidation of chlorpromazine and related phenothiazines. Cation radicals as the reactive intermediates in sulfoxide formation Eric Bosch and Jay K. Kochi pg 1057; DOI: 10.1039/P19950001057 |
Tandem sequence of ArSCl initiated AdE reactions resulting in formation of two C–C bonds Irina P. Smoliakova Ron Caple Vincent R. Magnuson Valery R. Polyakov William A. Smit Alexander S. Shashkov and Bato D. Ohinov pg 1065; DOI: 10.1039/P19950001065 |
Synthesis of the building blocks N-Fmoc-O-[-D-Ac3GalN3p-(1 Sandrine Rio-Anneheim Hans Paulsen Morten Meldal and Klaus Bock pg 1071; DOI: 10.1039/P19950001071 |
Conference diary pg viie; DOI: 10.1039/P1995000viie |
Front cover pg X033; DOI: 10.1039/P199500FX033 |
Journals bulletin pg X035; DOI: 10.1039/P1995000X035 |
Back cover pg X039; DOI: 10.1039/P199500BX039 |
Contents pages pg P097; DOI: 10.1039/P199500FP097 |
Back matter pg P105; DOI: 10.1039/P199500BP105 |
Potent inhibitor of the human rhinovirus (HRV) 3C protease containing a backbone modified glutamine Hing L. Sham William Rosenbrook Warren Kati David A. Betebenner Norman E. Wideburg Ayda Saldivar Jacob J. Plattner and Daniel W. Norbeck pg 1081; DOI: 10.1039/P19950001081 |
The behaviour of the furazan-N-methanide analogue of the furoxan system. Ring expansion: new routes to 6H-1,2,5-oxadiazines. A combined experimental and theoretical study Richard N. Butler Karen M. Daly John M. McMahon and Luke A. Burke pg 1083; DOI: 10.1039/P19950001083 |
Efficient regiospecific synthesis of two cytotoxic furonaphthoquinones, 5,7-dimethoxy-4,9-dihydronaphtho[2,3-b]furan-4,9-dione and 5,6,7-trimethoxy-4,9-dihydronaphtho[2,3-b]furan-4,9-dione Philip J. Perry Vasilios H. Pavlidis John A. Hadfield and Ian G. C. Coutts pg 1085; DOI: 10.1039/P19950001085 |
Simple synthetic approach to 6-oxa steroids. Synthesis of 6-oxa-5-pregnane-3,20-dione Daniel Nicoletti Alberto A. Ghini Adriana L. Brachet-Cota and Gerardo Burton pg 1089; DOI: 10.1039/P19950001089 |
S-Phenylacetamidomethyl (Phacm): an orthogonal cysteine protecting group for Boc and Fmoc solid-phase peptide synthesis strategies Miriam Royo Jordi Alsina Ernest Giralt Urszula Slomcyznska and Fernando Albericio pg 1095; DOI: 10.1039/P19950001095 |
Synthesis of novel inhibitors of electron transport G. Stuart Cockerill Philip C. Levett and Donald A. Whiting pg 1103; DOI: 10.1039/P19950001103 |
Synthesis of pyrrolidin-2-ones by 5-endo-trigonal radical cyclisation of N-vinyl-2,2-bis(phenylsulfanyl)acetamides Tatsunori Sato Noriko Chono Hiroyuki Ishibashi and Masazumi Ikeda pg 1115; DOI: 10.1039/P19950001115 |
Penitremones A–C, Penicillium metabolites containing an oxidised penitrem carbon skeleton giving insight into structure–tremorgenic relationships Jyotigna T. Naik Peter G. Mantle Richard N. Sheppard and Eric S. Waight pg 1121; DOI: 10.1039/P19950001121 |
Cyclopenta[b]indoles. Part 1. Synthesis of cyclopenta[b]indoles by formal [3 + 2] addition of indolylmethyl cations to alkenes Carrie-Ann Harrison Ralf Leineweber Christopher J. Moody and Jonathan M. J. Williams pg 1127; DOI: 10.1039/P19950001127 |
Cyclopenta[b]indoles. Part 2. Model studies towards the tremorgenic mycotoxins Carrie-Ann Harrison P. Mark Jackson Christopher J. Moody and Jonathan M. J. Williams pg 1131; DOI: 10.1039/P19950001131 |
Preparation of oxonanes and azonanes by oxidative ring expansion: synthesis of obtusan David S. Brown Mark C. Elliott Christopher J. Moody and Timothy J. Mowlem pg 1137; DOI: 10.1039/P19950001137 |
New syntheses of arylphosphinic acids from the reaction of ethyl diethoxymethylphosphinate with aryl bromides and phenols Stuart N. L. Bennett and Roger G. Hall pg 1145; DOI: 10.1039/P19950001145 |
Hydrocyanation of some ,-unsaturated ketones, and the synthesis of some unusual isoxazoles Wesley Cocker David H. Grayson and Patrick V. R. Shannon pg 1153; DOI: 10.1039/P19950001153 |
Synthesis of fluorescent derivatives of 3-O-(6-aminohexanoyl)pyrimidine nucleosides 5-triphosphates that act as DNA polymerase substrates reversibly tagged at C-3 Robert S. Sarfati Thomas Berthod Catherine Guerreiro and Bruno Canard pg 1163; DOI: 10.1039/P19950001163 |
Synthesis of the potent influenza neuraminidase inhibitor 4-guanidino Neu5Ac2en. X-Ray molecular structure of 5-acetamido-4-amino-2,6-anhydro-3,4,5-trideoxy-D-erythro-L-gluco-nononic acid Malcolm Chandler Mark J. Bamford Richard Conroy Brian Lamont Bina Patel Vipulkumar K. Patel Ian P. Steeples Richard Storer Niall G. Weir Michael Wright and Christopher Williamson pg 1173; DOI: 10.1039/P19950001173 |
Synthesis of 6-, 7- and 8-carbon sugar analogues of potent anti-influenza 2,3-didehydro-2,3-dideoxy-N-acetylneuraminic acid derivatives Mark J. Bamford Julia Castro Pichel Wahid Husman Bina Patel Richard Storer and Niall G. Weir pg 1181; DOI: 10.1039/P19950001181 |
Approaches to carbocyclic analogues of the potent neuraminidase inhibitor 4-guanidino-Neu5Ac2en. X-Ray molecular structure of N-[(1S,2S,6R)-2-azido-6-benzyloxymethyl-4-formylcyclohex-3-enyl]acetamide Malcolm Chandler Richard Conroy Anthony W. J. Cooper R. Brian Lamont Jan J. Scicinski James E. Smart Richard Storer Niall G. Weir Richard D. Wilson and Paul G. Wyatt pg 1189; DOI: 10.1039/P19950001189 |
Corrigenda M. Cavazza G. Guella L. Nucci F. Pergola N. Bicchierini F. Pietra Takumi Oshima Kazushi Tamada Toshikazu Nagai Hiroshi Suginome Takahiko Kondoh Camelia Gogonea Vishwakarma Singh Hitoshi Got and Eiji sawa pg 1199; DOI: 10.1039/P19950001199 |
Conference diary pg viif; DOI: 10.1039/P1995000viif |
Front cover pg X041; DOI: 10.1039/P199500FX041 |
Back cover pg X043; DOI: 10.1039/P199500BX043 |
Contents pages pg P111; DOI: 10.1039/P199500FP111 |
Back matter pg P119; DOI: 10.1039/P199500BP119 |
Conversion of one enantiomer of the carbocyclic nucleoside synthon 2-azabicyclo[2.2.1]hept-5-en-3-one into the other Christopher F. Palmer and Raymond McCague pg 1201; DOI: 10.1039/P19950001201 |
Synthesis of pyrazole fatty ester derivatives in water: a sonochemical approach Marcel S. F. Lie Ken Jie and Prabhavathi Kalluri pg 1205; DOI: 10.1039/P19950001205 |
Preparation and reactions of lithium indolyl(dimethyl)zincates Yoshinori Kondo Nobuo Takazawa Akihiro Yoshida and Takao Sakamoto pg 1207; DOI: 10.1039/P19950001207 |
Synthesis of 3-hydroxythiophenes and thiophen-3(2H)-ones by pyrolysis of alkylsulfanylmethylene Meldrum's acid derivatives Gordon A. Hunter and Hamish McNab pg 1209; DOI: 10.1039/P19950001209 |
Pigments of fungi. Part 41. Synthesis of (S)-(+)- and ()-dermolactone; stereochemistry of dermolactone from the Australian fungus Dermocybe sanguinea(Wulf. ex Fr.) Wnsche sensu Cleland Ann S. Cotterill Melvyn Gill and Nives M. Milanovic pg 1215; DOI: 10.1039/P19950001215 |
Some pyrrolopyrimidine chemistry directed to the synthesis of tricyclic purine analogues David M. Williams and Daniel M. Brown pg 1225; DOI: 10.1039/P19950001225 |
Chemistry of the mycalamides, antiviral and antitumour compounds from a marine sponge. Part 5. Acid-catalysed hydrolysis and acetal exchange, double bond additions and oxidation reactions Andrew M. Thompson John W. Blunt Murray H. G. Munro and Nigel B. Perry pg 1233; DOI: 10.1039/P19950001233 |
On the reaction between 3-bromo-2-nitrobenzo[b]thiophene and some amines: a novel aromatic nucleophilic substitution with rearrangement Francesco Guerrera Loredana Salerno Liliana Lamartina and Domenico Spinelli pg 1243; DOI: 10.1039/P19950001243 |
Synthesis of enantiomerically pure (R)- and (S)-2-sulfanylpropanoic acids (thiolactic acid) from ethyl (S)-lactate using pig liver esterase Robert P. Hof and Richard M. Kellogg pg 1247; DOI: 10.1039/P19950001247 |
Synthesis of all four diastereoisomers of 4-(carboxymethyl)proline, a conformationally constrained analogue of 2-aminoadipic acid Roberto Pellicciari Loredana Arenare Paolo De Caprariis Benedetto Natalini Maura Marinozzi and Alessandro Galli pg 1251; DOI: 10.1039/P19950001251 |
Dimethyl 3-chloroprop-1-en-2-ylphosphonate. Part 2. Alkylation of amines, phosphines and phosphites Igor E. Gurevich and John C. Tebby pg 1259; DOI: 10.1039/P19950001259 |
Directed lithiation of unprotected benzoic acids Bernard Bennetau Jacques Mortier Joël Moyroud and Jean-Luc Guesnet pg 1265; DOI: 10.1039/P19950001265 |
Synthesis of ()-[4a,4b,10b,12a]-9-halogeno-2-methyl-1,2,3,4,4a,4b,5,6,10b,11,12,12a-dodecahydronaphtho[2,1-]isoquinolines Graham L. Patrick pg 1273; DOI: 10.1039/P19950001273 |
Stereocontrol in cyclisation of dioxolanyl radicals Andrei S. Batsanov Michael J. Begley Rodney J. Fletcher John A. Murphy and Michael S. Sherburn pg 1281; DOI: 10.1039/P19950001281 |
Biocatalytic preparation of chiral alcohols by enantioselective reduction with immobilized cells of carrot Yoshihiko Akakabe Mirai Takahashi Makoto Kamezawa Keiichi Kikuchi Hojun Tachibana Takehiko Ohtani and Yoshinobu Naoshima pg 1295; DOI: 10.1039/P19950001295 |
Medium-sized cyclophanes. Part 36. Synthesis and conformational studies of dimethoxy[m.n]metacyclophanes Takehiko Yamato Jun-ichi Matsumoto Mitsuhiro Sato Kozo Noda and Masashi Tashiro pg 1299; DOI: 10.1039/P19950001299 |
Bromination–dehydrobromination route to some naturally occurring 1,6-dioxaspiro[4.4]-nonenes and -nonadienes Yong Qiang Tu Karl A. Byriel Colin H. L. Kennard and William Kitching pg 1309; DOI: 10.1039/P19950001309 |
Synthesis of N-aminomethylpyrrolidin-2-ones Ping Chen Dong-Jin Suh and Michael B. Smith pg 1317; DOI: 10.1039/P19950001317 |
Photochromic heterocyclic fulgides. Part 8. The condensation of 2,6-dichlorobenzaldehyde with diethyl [1-(2,5-dimethyl-3-furyl)ethylidene]succinate to give 6-chloro-2-(2,5-dimethyl-3-furyl)-1H-benzocycloheptene-3,4-dicarboxylic anhydride and photochromic (7S,7aS)-7-(2,6-dichlorophenyl)-2,4,7a-trimethyl-7,7a-dihydrobenzofuran-5,6-dicarboxylic anhydride Harry G. Heller Christopher J. Morgan and Matthew J. Ottaway pg 1323; DOI: 10.1039/P19950001323 |
Conference diary pg viig; DOI: 10.1039/P1995000viig |
Front cover pg X045; DOI: 10.1039/P199500FX045 |
Back cover pg X047; DOI: 10.1039/P199500BX047 |
Contents pages pg P121; DOI: 10.1039/P199500FP121 |
Back matter pg P129; DOI: 10.1039/P199500BP129 |
Electrochemical fluorination of 4-trimethylsilylazetidin-2-ones: an efficient and regioselective preparation of 4-fluoroazetidin-2-ones Kohji Suda Katsumi Hotoda Mitsuaki Aoyagi and Toshikatsu Takanami pg 1327; DOI: 10.1039/P19950001327 |
A direct and stereoselective route to (Z)-2-iodoalk-2-enes via-oxido phosphonium ylides Yanchang Shen and Shu Gao pg 1331; DOI: 10.1039/P19950001331 |
Phosphoramidate mediated conversion of tricarbonyl(vinylketene)iron(0) complexes into tricarbonyl(vinylketenimine)iron(0) complexes Stephen A. Benyunes Susan E. Gibson (née Thomas) and James A. Stern pg 1333; DOI: 10.1039/P19950001333 |
Potential mechanism-based tyrosine kinase inhibitors. Part 2. Design and synthesis of peptides containing heterocyclic tyrosine analogues David M. Andrews Mary Gregoriou Timothy C. M. Page Josephine M. Peach and Andrew J. Pratt pg 1335; DOI: 10.1039/P19950001335 |
The squalestatins: cleavage of the bicyclic core via the novel 6,8-dioxabicyclo[3.2.1]octane ring system Panayiotis A. Procopiou Esme J. Bailey Chuen Chan Graham G. A. Inglis Michael G. Lester Anton R. P. Srikantha Philip J. Sidebottom and Nigel S. Watson pg 1341; DOI: 10.1039/P19950001341 |
Trapping of translocated radicals by tetrathiafulvalene radical cation John A. Murphy and Stephen J. Roome pg 1349; DOI: 10.1039/P19950001349 |
SN2 Ring opening of aziridines bearing an ,-unsaturated ester group with organocopper reagents. A new stereoselective synthetic route to (E)-alkene dipeptide isosteres Nobutaka Fujii Kazuo Nakai Hirokazu Tamamura Akira Otaka Norio Mimura Yoshihisa Miwa Tooru Taga Yoshinori Yamamoto and Toshiro Ibuka pg 1359; DOI: 10.1039/P19950001359 |
Chemoselectivity and stereoselectivity of cyclisation of -diazocarbonyls leading to oxygen and sulfur heterocycles catalysed by chiral rhodium and copper catalysts Tao Ye Concepción Fernández García and M. Anthony McKervey pg 1373; DOI: 10.1039/P19950001373 |
Reactions of tosyl azide with 2-phenoxy- and 2-phenylsulfanyl-2,3-dihydro-1H-indane-1,3-dione. Unexpected reactivity of intermediate 4-acyl-5-hydroxy-1-tosyltriazolines Luisa Benati Gianluca Calestani Pier Carlo Montevecchi and Piero Spagnolo pg 1381; DOI: 10.1039/P19950001381 |
Synthesis of 4-thia-2-azapodophyllotoxin, a new analogue of the antitumour lignan podophyllotoxin Yukio Hitotsuyanagi Masatsugu Kobayashi Koichi Takeya and Hideji Itokawa pg 1387; DOI: 10.1039/P19950001387 |
Approach to the synthesis of 4-demethylforskolin (19-norforskolin) Jerry J. Harnett James K. Sutherland and Hua Yang pg 1391; DOI: 10.1039/P19950001391 |
The chemoselective cyclisation of unsymmetrical -diketones to cyclopentenones by directed aldol reaction using a magnesium chelate Michael L. F. Cadman Leslie Crombie Stephen Freeman and Jayshree Mistry pg 1397; DOI: 10.1039/P19950001397 |
Dioxolane nucleosides and their phosphonate derivatives: synthesis and hydrolytic stability Ekaterina V. Efimtseva Sergey N. Mikhailov Sergey Meshkov Teemu Hankamäki Mikko Oivanen and Harri Lönnberg pg 1409; DOI: 10.1039/P19950001409 |
Synthesis of novel carbo- and heteropolycycles. Part 30. 1,3-Dipolar cycloaddition of nitrile functions with some selected nitrones. Efficient synthesis of 2,3-dihydro-1,2,4-oxadiazole derivatives Yang Yu Naoto Watanabe Masatomi Ohno and Shoji Eguchi pg 1417; DOI: 10.1039/P19950001417 |
Asymmetric reduction of a carbon–nitrogen double bond: enantioselective synthesis of 4,5-dihydro-3H-2,3-benzodiazepines István Ling Benjamin Podányi Tamás Hámori and Sándor Sólyom pg 1423; DOI: 10.1039/P19950001423 |
Synthesis of azophenolic crown ethers of Cs symmetry incorporating cis-1-phenylcyclohexane-1,2-diol residues as a steric barrier and diastereotopic face selectivity in complexation of amines by their diastereotopic faces Koichiro Naemura Sachiko Takeuchi Masaki Asada Koji Ueno Keiji Hirose Yoshito Tobe Takahiro Kaneda and Yoshiteru Sakata pg 1429; DOI: 10.1039/P19950001429 |
Furan-2(3H)- and -2(5H)-ones. Part 6. Di--methane rearrangement of the -substituted 4-benzylfuran-2(5H)-one system Osamu Muraoka Genzoh Tanabe Mié Higashiura Toshie Minematsu and Takefumi Momose pg 1437; DOI: 10.1039/P19950001437 |
Studies on fused pyrimidine derivatives. Part 14. Formation and transformation of [4 + 2] cycloadducts, cyclohepta[g]quinazoline derivatives, by the reaction of 5-(arylaminomethylene)-1,3-dimethyl-6-methyleneperhydropyrimidine-2,4-diones with tropone Ken Ikuno Takashi Kobayashi Toshio Harada Michihiko Noguchi and Akikazu Kakehi pg 1445; DOI: 10.1039/P19950001445 |
Studies on fused pyrimidine derivatives. Part 15. Features and mechanistic considerations of the reaction of 5-(alkylaminomethylene)-6-methyleneperhydropyrimidine-2,4-diones with tropone Takashi Kobayashi Ken Ikuno Michihiko Noguchi and Akikazu Kakehi pg 1453; DOI: 10.1039/P19950001453 |
Photocleavage of the C–O bond of 9-phenanthrylmethyl -anilinoalkyl ethers via photo-induced intramolecular electron transfer Akira Sugimoto Satoshi Kimoto Tomohiro Adachi and Hiroo Inoue pg 1459; DOI: 10.1039/P19950001459 |
Conference diary pg viih; DOI: 10.1039/P1995000viih |
Front cover pg X049; DOI: 10.1039/P199500FX049 |
Back cover pg X051; DOI: 10.1039/P199500BX051 |
Contents pages pg P133; DOI: 10.1039/P199500FP133 |
Back matter pg P143; DOI: 10.1039/P199500BP143 |
Enantiocomplementary asymmetric epoxidation of selected enones using poly-L-leucine and poly-D-leucine M. Elena Lasterra Sánchez and Stanley M. Roberts pg 1467; DOI: 10.1039/P19950001467 |
1,4-Asymmetric induction in reactions between [2-(1-alkoxyalkyl)propenyl](tributyl)stannanes and aldehydes promoted by tin(IV) halides Michelangelo Gruttadauria and Eric J. Thomas pg 1469; DOI: 10.1039/P19950001469 |
Nucleophilic aromatic substitution of 2-sulfonyl-substituted 1-methoxynaphthalenes with Grignard reagents Tetsutaro Hattori Mikio Suzuki Yasuko Komuro and Sotaro Miyano pg 1473; DOI: 10.1039/P19950001473 |
Azoles. Part II. Synthesis of imidazole-2(and -5)-carbaldehydes and derivatives of imidazo[1,2-b]isoquinoline; transmetallation of imidazol-5-yllithium compounds Brian Iddon Anders K. Petersen Jan Becher and Nils J. Christensen pg 1475; DOI: 10.1039/P19950001475 |
Synthesis and biological activity of new C-6 and C-7 substituted vinyloxyimino-penicillins and -cephalosporins Stephen C. M. Fell Michael J. Pearson George Burton and John S. Elder pg 1483; DOI: 10.1039/P19950001483 |
Synthesis of secasterone and further epimeric 2,3- epoxybrassinosteroids Brunhilde Voigt Suguru Takatsuto Takao Yokota and Günter Adam pg 1495; DOI: 10.1039/P19950001495 |
Conversion of benzene and chlorobenzene into polyhydroxylated cyclohexane derivatives related to cyclophellitol Stanley M. Roberts and Peter W. Sutton pg 1499; DOI: 10.1039/P19950001499 |
Enzymatic Baeyer–Villiger oxidations of some bicyclo[2.2.1]heptan-2-ones using monooxygenases from Pseudomonas putida NCIMB 10007: enantioselective preparation of a precursor of azadirachtin René Gagnon Gideon Grogan Stanley M. Roberts Raffaella Villa and Andrew J. Willetts pg 1505; DOI: 10.1039/P19950001505 |
Synthesis and the absolute configuration of the sesquiterpene aldehyde tridensenal from the Taiwanese liverwort Bazzania tridens Motoo Tori Naomi Uchida Aya Sumida Hirosuke Furuta and Yoshinori Asakawa pg 1513; DOI: 10.1039/P19950001513 |
1H and 13C NMR characterization of new oleuropein aglycones Rita Limiroli Roberto Consonni Gianluca Ottolina Vincenzo Marsilio Giorgio Bianchi and Lucia Zetta pg 1519; DOI: 10.1039/P19950001519 |
Synthesis of vinylsilanes by silyl-cupration of acetylenes using tert-butyldiphenylsilyl-cuprate reagents Asunción Barbero Purificación Cuadrado Ian Fleming Ana M. González Francisco J. Pulido and Alicia Sánchez pg 1525; DOI: 10.1039/P19950001525 |
Reactions of cyclic -keto esters and other enol derivatives with 3-acetoxyamino-2-isopropylquinazolin-4(3H)-one: further oxidation of the cyclic -(3,4-dihydro-2-isopropyl-4-oxoquinazolin-3-yl)amino ketones with lead tetraacetate leading to ring-expansion (in dichloromethane) and ring-cleavage (in methanol) Robert S. Atkinson Emma Barker Paul J. Edwards and Gordon A. Thomson pg 1533; DOI: 10.1039/P19950001533 |
Total synthesis of 2-deoxy-2-arafluoro-tubercidin, -toyocamycin, -sangivamycin and certain related nucleosides Birendra K. Bhattacharya T. Sudhakar Rao and Ganapathi R. Revankar pg 1543; DOI: 10.1039/P19950001543 |
Total synthesis of (–)-ovalicin and analogues from L-quebrachitol Derek H. R. Barton Sophie Bath David C. Billington Stephan D. Gero Béatrice Quiclet-Sire and Mohammad Samadi pg 1551; DOI: 10.1039/P19950001551 |
Stereoselective syntheses of D-ribo- and L-lyxo-phytosphingosine Yun-Long Li Xiu-Hong Mao and Yu-Lin Wu pg 1559; DOI: 10.1039/P19950001559 |
Biosynthesis of violacein: oxygenation at the 2-position of the indole ring and structures of proviolacein, prodeoxyviolacein and pseudoviolacein, the plausible biosynthetic intermediates of violacein and deoxyviolacein Tsutomu Hoshino Toru Hayashi and Taro Odajima pg 1565; DOI: 10.1039/P19950001565 |
2-Deoxy-2-trichloroacetamido-D-glucopyranose derivatives in oligosaccharide synthesis: from hyaluronic acid to chondroitin 4-sulfate trisaccharides Caroline Coutant and Jean-Claude Jacquinet pg 1573; DOI: 10.1039/P19950001573 |
Ring transformation of the adducts of the polar cycloadditions of 2-benzothiopyrylium salts Hiroshi Shimizu Shojiro Miyazaki Tadashi Kataoka and Mikio Hori pg 1583; DOI: 10.1039/P19950001583 |
Direct visualization of enzyme inhibitors using a portion mixing inhibitor library containing a quenched fluorogenic peptide substrate. Part 1. Inhibitors for subtilisin Carlsberg Morten Meldal and Ib Svendsen pg 1591; DOI: 10.1039/P19950001591 |
Formation of polycyclic compounds in the photoreactions of 9-(-anilinoalkyl)phenanthrenes Akira Sugimoto Noriyuki Fukada Tomohiro Adachi and Hiroo Inoue pg 1597; DOI: 10.1039/P19950001597 |
Synthesis of L-threo- and L-erythro-[1-13C, 2,3-2H2]amino acids: novel probes for conformational analysis of peptide side chains Makoto Oba Ryuichi Ueno Mika Fukuoka (née Yoshida) Masatsune Kainosho and Kozaburo Nishiyama pg 1603; DOI: 10.1039/P19950001603 |
Synthesis and lyotropic phase behaviour of methyl 3,4-di-O-hexyl- and -di-O-octyl--lactoside and partial O-acetylation of methyl 3,4-di-O-octyl--lactoside Virginie Langlois and J. Michael Williams pg 1611; DOI: 10.1039/P19950001611 |
Synthesis of partial nonpeptidic peptide mimetics as potential neurotensin agonists and antagonists Alan P. Kozikowski Dharmpal S. Dodd Javid Zaidi Yuan-Ping Pang Bernadette Cusack and Elliott Richelson pg 1615; DOI: 10.1039/P19950001615 |
Synthetic studies on morphine-based analgesics. Intramolecular Diels–Alder approach to 4a-aryldecahydroisoquinolines Sheetal Handa Keith Jones and Christopher G. Newton pg 1623; DOI: 10.1039/P19950001623 |
Alternative synthesis of 2-arylpropanoic acids from enolate and aryl halides Carlos G. Ferrayoli Sara M. Palacios and Rubén A. Alonso pg 1635; DOI: 10.1039/P19950001635 |
Conference diary pg ixa; DOI: 10.1039/P19950000ixa |
Front cover pg X053; DOI: 10.1039/P199500FX053 |
Back cover pg X055; DOI: 10.1039/P199500BX055 |
Contents pages pg P145; DOI: 10.1039/P199500FP145 |
Back matter pg P153; DOI: 10.1039/P199500BP153 |
A new approach to the synthesis of dipeptides with unnatural amino acids using organozinc chemistry Michael J. Dunn Sylvie Gomez and Richard F. W. Jackson pg 1639; DOI: 10.1039/P19950001639 |
Oxidation of methyl p-tolyl sulfide with bakers' yeast: preparation of a synthon of the mevinic acid-type hypocholestemic agents Jean Beecher Ian Brackenridge Stanley M. Roberts Jenny Tang and Andrew J. Willetts pg 1641; DOI: 10.1039/P19950001641 |
Lipase-promoted asymmetric transesterification of 4-alkyloxetan-2-ones with ring-opening Yota Koichi Kaoru Suginaka and Yukio Yamamoto pg 1645; DOI: 10.1039/P19950001645 |
Ring expansion reactions of isoquinoline derivatives to 2-benzazocine and 3-benzazecine derivatives Mostafa M. M. Bamatraf John M. Vernon and Giles D. Wilson pg 1647; DOI: 10.1039/P19950001647 |
A phenanthrolinoquinomethane: synthesis and study of precursors Noemie Fixler Hervé Salez Martine Demeunynck and Jean Lhomme pg 1649; DOI: 10.1039/P19950001649 |
Reactions of N-sulfinylarylamines with 1,4-benzoquinone and 1,4-naphthoquinone: synthesis of N-aryl sulfinamoyl quinones and their hydrolysis to hydroxyquinones Ananda S. Amarasekara and W. Wimal Pathmasiri pg 1653; DOI: 10.1039/P19950001653 |
Some chemistry of 4,5-dichloro-1,2,3-dithiazolium chloride and its derivatives Thierry Besson and Charles W. Rees pg 1659; DOI: 10.1039/P19950001659 |
Biosynthesis of aspinonene, a branched pentaketide produced by Aspergillus ochraceus, related to aspyrone Jens Fuchser Ralf Thiericke and Axel Zeeck pg 1663; DOI: 10.1039/P19950001663 |
Synthesis and use of (E)-1-ethoxy-3-fluoroalkyl-3-hydroxy-4-(4-methylphenylsulfinyl)but-1-enes Pierfrancesco Bravo Luca Bruché Alessandra Farina Igor I. Gerus Maria T. Kolytcheva Valery P. Kukhar Stefano Valdo Meille and Fiorenza Viani pg 1667; DOI: 10.1039/P19950001667 |
Parasite glycoconjugates. Part 3. Synthesis of substrate analogues of early intermediates in the biosynthetic pathway of glycosylphosphatidylinositol membrane anchors Sylvain Cottaz John S. Brimacombe and Michael A. J. Ferguson pg 1673; DOI: 10.1039/P19950001673 |
Organolead-mediated arylation of allyl -keto esters: selective synthesis of 2-hydroxyisoflavones Dervilla M. X. Donnelly Jean-Pierre Finet and Bernard A. Rattigan pg 1679; DOI: 10.1039/P19950001679 |
Synthesis of S-alkyl esters of protected 2-deoxyribonucleoside 3-phosphorothioates. Building blocks for the large-scale synthesis of phosphorothioate analogues of oligodeoxyribonucleotides by the phosphotriester approach in solution Xiaohai Liu and Colin B. Reese pg 1685; DOI: 10.1039/P19950001685 |
Preparation of optically active derivatives of (1,4/2,3,5)- and (1,2,3,4,5/0)-5-aminocyclopentane-1,2,3,4-tetraols: synthesis of mannostatin A and its enantiomer Seiichiro Ogawa Hiroshi Kimura Chikara Uchida and Takashi Ohashi pg 1695; DOI: 10.1039/P19950001695 |
Synthesis of trehazolin analogues containing modified sugar moieties Chikara Uchida Hideo Kitahashi Shinsuke Watanabe and Seiichiro Ogawa pg 1707; DOI: 10.1039/P19950001707 |
New synthesis of hypervalent T-shaped coordination compounds of selenium by the reaction of bis(2-bromoethyl)selenium dibromide with pyridine and its derivatives Masatsugu Miura Yoshinori Takanohashi Yoichi Habata and Sadatoshi Akabori pg 1719; DOI: 10.1039/P19950001719 |
Cuprous bromide-promoted cyclization of ketene N,S-acetals with prop-2-ynyl bromide: synthesis of regiospecifically substituted and annelated 3-acyl(or nitro)-5-methyl pyrroles Akhilesh K. Gupta Kethiri R. Reddy Hiriyakkanavar Ila and Hiriyakkanavar Junjappa pg 1725; DOI: 10.1039/P19950001725 |
Addition–cyclization of a diallylmalonic acid ester and related compounds with per(poly)fluoroalkyl iodides using a trichlorolanthanide [LnCl3(cat.)]/Zn system Wei-Yuan Huang Gang Zhao and Yu Ding pg 1729; DOI: 10.1039/P19950001729 |
Strong inhibitory effect of sugarbiphenylylboronic acid complexes on the hydrolytic activity of -chymotrypsin Hikaru Suenaga Masafumi Mikami Hiromasa Yamamoto Takaaki Harada and Seiji Shinkai pg 1733; DOI: 10.1039/P19950001733 |
Synthesis of major histocompatibility complex class I binding glycopeptides Gemma Arsequell John S. Haurum Tim Elliott Raymond A. Dwek and Annemarie C. Lellouch pg 1739; DOI: 10.1039/P19950001739 |
Synthesis of tetrazoles bearing a sugar moiety (sugar tetrazoles). X-Ray molecular structure of (7R,8R,9S,10R)-8,9,10-tribenzyloxy-7-benzyloxymethyl-6-oxa-1,5-pentamethylenetetrazole Masataka Yokoyama Sachiko Hirano Michio Matsushita Takeshi Hachiya Naoki Kobayashi Misao Kubo Hideo Togo and Hiroko Seki pg 1747; DOI: 10.1039/P19950001747 |
New digitalis steroids. Synthesis of 17-amino 5,14-steroids by thermolysis of 17-azidocarbonyloxymethyl derivatives Giorgio Fedrizzi Luigi Bernardi Giuseppe Marazzi Piero Melloni and Marco Frigerio pg 1755; DOI: 10.1039/P19950001755 |
Diels–Alder reaction of benzylidene(cyano)methyl-1,3-benzoxa/thiazoles as stable 1-azabuta-1,3-dienes Masanori Sakamoto Asae Nozaka Mino Shimamoto Hideki Ozaki Yoko Suzuki Sanae Yoshioka Mayumi Nagano Kimio Okamura Tadamasa Date and Osamu Tamura pg 1759; DOI: 10.1039/P19950001759 |
Synthesis of ,-disubstituted acetic acids using low-valent titanium Mariano García Carmen del Campo Emilio F. Llama and José V. Sinisterra pg 1771; DOI: 10.1039/P19950001771 |
3,4-Di-O-methylcedrusin: synthesis, resolution and absolute configuration Guy Lemière Mei Gao Alex De Groot Roger Dommisse Josef Lepoivre Luc Pieters and Volker Buss pg 1775; DOI: 10.1039/P19950001775 |
Corrigendum Jim-Min Fang Chun-Hung Lin Curt W. Bradshaw and Chi-Huey Wong pg 1781; DOI: 10.1039/P19950001781 |
Conference diary pg viii; DOI: 10.1039/P1995000viii |
Front cover pg X057; DOI: 10.1039/P199500FX057 |
Back cover pg X059; DOI: 10.1039/P199500BX059 |
Contents pages pg P155; DOI: 10.1039/P199500FP155 |
Back matter pg P163; DOI: 10.1039/P199500BP163 |
Synthesis of the 1,4-diazepan-2-one moiety of liposidomycins Kwan Soo Kim In Haeng Cho Yeong Hee Ahn and Jong Il Park pg 1783; DOI: 10.1039/P19950001783 |
Synthesis and X-ray crystal structure of 1,3,5-tris(fluoren-9-ylidenemethyl)benzene: towards a C48-fragment of [60]-fullerene Goverdhan Mehta K. Venkateswara Rao and K. Ravikumar pg 1787; DOI: 10.1039/P19950001787 |
The inverse electron-demand Diels–Alder reaction in polymer synthesis. Part 2. Some bis(1,2,4-triazines) as potential bis-diene monomers Michael J. Bruce Gillian A. McLean Brodyck J. L. Royles David M. Smith and Paul N. Standring pg 1789; DOI: 10.1039/P19950001789 |
Anthraquinone-photocatalysed addition of amines to ,-unsaturated esters: a novel route to indolizidone, pyrrolizidone and related ring systems Suresh Das J. S. Dileep Kumar K. Shivaramayya and M. V. George pg 1797; DOI: 10.1039/P19950001797 |
Synthesis of bridged azabicyclic compounds using radical translocation reactions of 1-(o-bromobenzoyl)-2-(prop-2-enyl)pyrrolidines Tatsunori Sato Yasuhiro Kugo Erina Nakaumi Hiroyuki Ishibashi and Masazumi Ikeda pg 1801; DOI: 10.1039/P19950001801 |
Docetaxel (taxotere) derivatives: novel NbCl3-based stereoselective approach to 2-methyldocetaxel Jean-Noël Denis Abdellatif Fkyerat Yves Gimbert Claire Coutterez Pierre Mantellier Sylvie Jost and Andrew E. Greene pg 1811; DOI: 10.1039/P19950001811 |
Synthesis and characterisation of some novel phthalocyanines containing both oligo(ethyleneoxy) and alkyl or alkoxy side-chains: novel unsymmetrical discotic mesogens Guy J. Clarkson Neil B. McKeown and Kevin E. Treacher pg 1817; DOI: 10.1039/P19950001817 |
The mechanism of directed remote asymmetric reduction of carbonyl groups via homochiral boronate esters Gráinne Conole Richard J. Mears Harshani De Silva and Andrew Whiting pg 1825; DOI: 10.1039/P19950001825 |
Alkylation of 6-N-acylated adenosine derivatives by the use of phase transfer catalysis Keiichi Aritomo Takeshi Wada and Mitsuo Sekine pg 1837; DOI: 10.1039/P19950001837 |
Titanium(IV) mediated reductive aminations of 1-adamantyl methyl ketone: facile preparation of potential antiviral agents rimantadine and its analogues Sukanta Bhattacharyya pg 1845; DOI: 10.1039/P19950001845 |
Antibiotic peptides from Trichoderma harzianum: harzianins HC, proline-rich 14-residue peptaibols Sylvie Rebuffat Christophe Goulard and Bernard Bodo pg 1849; DOI: 10.1039/P19950001849 |
Intramolecular 1,3-dipolar cycloaddition at the periphery of heterocyclic systems. Part 1. Facile oxime–nitrone isomerisation at the periphery of pyran and 1-benzopyran Mitsuhiro Gotoh Takahiro Mizui Bin Sun Ken Hirayama and Michihiko Noguchi pg 1857; DOI: 10.1039/P19950001857 |
Asymmetric Diels–Alder reactions between chiral sugar nitroalkenes and 1-O-substituted buta-1,3-dienes. Synthesis and reactivity of new cyclohexenyl derivatives José A. Serrano Luis E. Cáceres and Emilio Román pg 1863; DOI: 10.1039/P19950001863 |
Synthesis, resolution and absolute configuration determination of (S)- and (R)-4-formyl-5-hydroxy [2.2]paracyclophane and its application in the asymmetric synthesis of -amino acids Dmitri Yu. Antonov Yuri N. Belokon Nikolai S. Ikonnikov Svetlana A. Orlova Aleksander P. Pisarevsky Nikolai I. Raevski Valeria I. Rozenberg Elena V. Sergeeva Yuri T. Struchkov Vitali I. Tararov and Evgeni V. Vorontsov pg 1873; DOI: 10.1039/P19950001873 |
Conference diary pg viij; DOI: 10.1039/P1995000viij |
Front cover pg X061; DOI: 10.1039/P199500FX061 |
Back cover pg X063; DOI: 10.1039/P199500BX063 |
Contents pages pg P165; DOI: 10.1039/P199500FP165 |
Back matter pg P173; DOI: 10.1039/P199500BP173 |
Cerium(IV) ammonium nitrate mediated addition of dimethyl malonate to styrene: a remarkable reaction Vijay Nair and Jessy Mathew pg 1881; DOI: 10.1039/P19950001881 |
Design and synthesis of a C4-symmetrical hard–soft ditopic metal receptor by calixarene–porphyrin coupling Takeshi Nagasaki Hiroyuki Fujishima Masayuki Takeuchi and Seiji Shinkai pg 1883; DOI: 10.1039/P19950001883 |
Selective mono-benzylation of methylene active compounds with dibenzyl carbonate: benzylation of phenol Maurizio Selva Carlos Alberto Marques and Pietro Tundo pg 1889; DOI: 10.1039/P19950001889 |
Carotenoids and related polyenes. Part 3. First total synthesis of fucoxanthin and halocynthiaxanthin using oxo-metallic catalyst Yumiko Yamano Chisato Tode and Masayoshi Ito pg 1895; DOI: 10.1039/P19950001895 |
Synthesis of DL-threo-3-(1-fluoro-1-methylethyl)- and DL-threo-3-(1,1-difluoroethyl)malic acids. Mechanistic studies of 3-isopropylmalate dehydrogenase Tetsuya Aoyama Tadashi Eguchi Tairo Oshima and Katsumi Kakinuma pg 1905; DOI: 10.1039/P19950001905 |
Control over absolute (R,S), relative (syn,anti) and geometrical (E,Z) stereochemistry in the synthesis of allylically substituted alkenes from diphenylphosphinoyl epoxy alcohols Jonathan Clayden Andrew B. McElroy and Stuart Warren pg 1913; DOI: 10.1039/P19950001913 |
Biosynthesis of (+)-cubenene and (+)-epicubenol by cell-free extracts of cultured cells of Heteroscyphus planus and cyclization of [2H]farnesyl diphosphates Kensuke Nabeta Kazuyoshi Kigure Masaru Fujita Tomomi Nagoya Takehiro Ishikawa Hiroshi Okuyama and Toshihide Takasawa pg 1935; DOI: 10.1039/P19950001935 |
Radical substitution on a thioester by a methyl radical generated from methyl(L)cobaloxime Masaru Tada Takao Yoshihara and Kiyohiko Sugano pg 1941; DOI: 10.1039/P19950001941 |
Synthesis of chiral diazanedicarboxylate and diazenedicarboxylate esters: electrophilic amination reactions of achiral ester and amide enolates Joanna M. Harris Evon A. Bolessa Aubrey J. Mendonca Sheng-Chu Feng and John C. Vederas pg 1945; DOI: 10.1039/P19950001945 |
Synthesis of macrocyclic diazanedicarboxylate and diazenedicarboxylate esters containing a steroid skeleton: an unusual oxidation of bromide to bromine by a strained diazenedicarboxylate ester. X-Ray molecular structure of 3-(3-hydroxypropyl)-24-nor-5-cholan-7-ol diazane-1,2-dicarboxylate cyclic diester Joanna M. Harris Evon A. Bolessa and John C. Vederas pg 1951; DOI: 10.1039/P19950001951 |
Electro-organic reactions. Part 42. The diastereoselective cathodic hydrodimerisation of cinnamate esters; preparative aspects James H. P. Utley Mustafa Güllü and Majid Motevalli pg 1961; DOI: 10.1039/P19950001961 |
New synthesis of carboxin and oxycarboxin pesticides: application to the preparation of their new analogues substituted at the C-2 methyl group Romualdo Caputo Carla Ferreri Annalisa Guaragna Giovanni Palumbo and Silvana Pedatella pg 1971; DOI: 10.1039/P19950001971 |
Corrigenda Mark J. Bamford Julia Castro Pichel Wahid Husman Bina Patel Richard Storer Niall G. Weir John A. Murphy and Stephen J. Romme pg 1975; DOI: 10.1039/P19950001975 |
Conference diary pg viik; DOI: 10.1039/P1995000viik |
Front cover pg X065; DOI: 10.1039/P199500FX065 |
Back cover pg X067; DOI: 10.1039/P199500BX067 |
Contents pages pg P177; DOI: 10.1039/P199500FP177 |
Back matter pg P185; DOI: 10.1039/P199500BP185 |
Parasite glycoconjugates. Part 4. Chemical synthesis of disaccharide and phosphorylated oligosaccharide fragments of Leishmania donovani antigenic lipophosphoglycan Andrey V. Nikolaev Trevor J. Rutherford Michael A. J. Ferguson and John S. Brimacombe pg 1977; DOI: 10.1039/P19950001977 |
Tripolar mesoionic compounds Shuki Araki Jiro Mizuya Naomitsu Aoyama and Yasuo Butsugan pg 1989; DOI: 10.1039/P19950001989 |
Synthesis of photoactivatable fluorescein derivatives bearing side chains with varying properties John E. T. Corrie and David R. Trentham pg 1993; DOI: 10.1039/P19950001993 |
Synthesis of phosphorothioate esters of L-phenyl-lactic acid as transition-state inhibitors of carboxypeptidase A Jacqueline M. Hill and Gordon Lowe pg 2001; DOI: 10.1039/P19950002001 |
Regio- and enantio-selective catalytic epoxidation of conjugated dienes Kaare G. Rasmussen Dorte S. Thomsen and Karl Anker Jørgensen pg 2009; DOI: 10.1039/P19950002009 |
Improved preparation of -amyloid(1–43): structural insight leading to optimised positioning of N-(2-hydroxy-4-methoxybenzyl)(Hmb) backbone amide protection Martin Quibell William G. Turnell and Tony Johnson pg 2019; DOI: 10.1039/P19950002019 |
Synthesis and cathodic cleavage of a set of substituted benzenesulfonamides including the corresponding tert-butyl sulfonylcarbamates: pKa of sulfonamides Barthélémy Nyasse Leif Grehn Ulf Ragnarsson Hernani L. S. Maia Luis S. Monteiro Ivo Leito Ilmar Koppel and Juta Koppel pg 2025; DOI: 10.1039/P19950002025 |
Isomerisation of 4-aryl-4-methylhex-5-en-2-ones to 5-aryl-4-methylhex-5-en-2-ones by an intramolecular ene-retro ene reaction sequence A. Srikrishna K. Krishnan S. Venkateswarlu and P. Praveen Kumar pg 2033; DOI: 10.1039/P19950002033 |
Chemistry of silyl thioketones. Part 8. Photo-induced cycloadditions of silyl thioketones with olefins Bianca Flavia Bonini Mauro Comes Franchini Mariafrancesca Fochi Germana Mazzanti Alfredo Ricci Paolo Zani and Binne Zwanenburg pg 2039; DOI: 10.1039/P19950002039 |
Preparation of alkyl- and aryl-amino[2H2]methylphosphinic acids Sylvie Berté-Verrando François Nief Carl Patois and Philippe Savignac pg 2045; DOI: 10.1039/P19950002045 |
Asymmetric synthesis of steroidal Trger's base analogues. X-Ray molecular structure of methyl 3,12-{6H,12H-5,11-methanodibenzo[b,f][1,5]diazocine-2,8-bisacetoxy}-5-cholan-24-oate Uday Maitra Braja Gopal Bag Photon Rao and Douglas Powell pg 2049; DOI: 10.1039/P19950002049 |
Model for the functional active site of Baeyer–Villigerases. X-Ray crystal data for (1S,2R,5R,8S,1R)-8-endo-benzoyloxy-N-(1-phenylethyl)bicyclo[3.3.0]octane-2-endo-carboxamide David R. Kelly Christopher J. Knowles Jassem G. Mahdi Michael A. Wright Ian N. Taylor David E. Hibbs Michael B. Hursthouse Adel K. Mish'al Stanley M. Roberts Peter W. H. Wan Gideon Grogan and Andrew J. Willetts pg 2057; DOI: 10.1039/P19950002057 |
Metabolites of the higher fungi. Part 28. Globoscinic acid and globoscin, a labile acid–lactone system from Xylaria globosa and Xylaria obovata Monilola Adeboya Raymond L. Edwards Thomas Laessøe Derek J. Maitland and Anthony S. J. Whalley pg 2067; DOI: 10.1039/P19950002067 |
Conference diary pg viil; DOI: 10.1039/P1995000viil |
Front cover pg X069; DOI: 10.1039/P199500FX069 |
Back cover pg X071; DOI: 10.1039/P199500BX071 |
Contents pages pg P187; DOI: 10.1039/P199500FP187 |
Regioselectivity in the nickel-catalysed coupling of cyclic carbonates of but-3-ene-1,2-diols with organoborates Ryo Mizojiri and Yuichi Kobayashi pg 2073; DOI: 10.1039/P19950002073 |
Synthesis and reactivity of tricarbonyl(indan-2-one)chromium(0) E. Lucy M. Cowton Susan E. Gibson (née Thomas) Michael J. Schneider and Mark H. Smith pg 2077; DOI: 10.1039/P19950002077 |
Ring-opening desulfurization of 1,2,3-thiadiazolium salts with N-nucleophiles Gerrit L'abbé Peggy Vossen Wim Dehaen and Suzanne Toppet pg 2079; DOI: 10.1039/P19950002079 |
Keynote article. Nickel catalysed coupling of allylamines and boronic acids Barry M. Trost and Michel D. Spagnol pg 2083; DOI: 10.1039/P19950002083 |
1,2,3-Dithiazoles and new routes to 3,1-benzoxazin-4-ones, 3,1-benzothiazin-4-ones and N-arylcyanothioformamides Thierry Besson Kumaraswamy Emayan and Charles W. Rees pg 2097; DOI: 10.1039/P19950002097 |
2-Alkoxy-3-oxoalkyl-tetrahydropyrans and -tetrahydrofurans: versatile intermediates in heterocyclic synthesis Pierre Duhamel Abdallah Deyine Gilles Dujardin Gérard Plé and Jean-Marie Poirier pg 2103; DOI: 10.1039/P19950002103 |
Two alternative conformational states of ,-dialkylglycyl-L-prolyl sequences governed by presence/absence of an NH group directly following the proline residue. X-Ray crystal and molecular structures of Boc-D-Iva-L-Pro-NHBzl and Boc-L-Iva-L-Pro-NHBzl Masao Kawai Yoshimasa Omori Hatsuo Yamamura Yasuo Butsugan Tooru Taga and Yoshihisa Miwa pg 2115; DOI: 10.1039/P19950002115 |
Preparation of -methoxyallylphosphonates and their conversion into 2-methoxyalka-1,3-dienes Kevin Fettes Leslie McQuire and Alistair W. Murray pg 2123; DOI: 10.1039/P19950002123 |
A potential photoaffinity probe for labelling the active site of aequorin: a photolabile coelenterazine analogue with a trifluoromethyldiazirine group Feng Qi Chen Jing Ling Zheng Takashi Hirano Haruki Niwa Yoshihiro Ohmiya and Mamoru Ohashi pg 2129; DOI: 10.1039/P19950002129 |
Reactivity of [bis(1-adamantylcarbonyloxy)iodo]arenes in substitution and addition reactions Hideo Togo Rie Taguchi Kentaro Yamaguchi and Masataka Yokoyama pg 2135; DOI: 10.1039/P19950002135 |
Synthesis and thermal decomposition of azidovinylbenzo[b]thiophenes Alessandro Degl'Innocenti Maria Funicello Patrizia Scafato Piero Spagnolo and Paolo Zanirato pg 2141; DOI: 10.1039/P19950002141 |
Synthesis and oxidation of the decarbonylated adducts generated from alkenes and tricarbonyl(vinylketene)iron(0) complexes Susan E. Gibson (née Thomas) Stephen P. Saberi Alexandra M. Z. Slawin Paul D. Stanley Mark F. Ward David J. Williams and Paul Worthington pg 2147; DOI: 10.1039/P19950002147 |
Carbon–carbon bond formation and reduction of aldehydes, ketones and acetals with silylated nucleophiles catalysed by tetracyanoethylene Tsuyoshi Miura and Yukio Masaki pg 2155; DOI: 10.1039/P19950002155 |
Formal total syntheses of (–)-oudemansins A, B and X based on a lipase-catalysed hydrolysis of an acetate Hiroyuki Akita Cheng Yu Chen and Shinji Nagumo pg 2159; DOI: 10.1039/P19950002159 |
Comparison of N-Dts and N-Aloc in the solid-phase syntheses of O-GlcNAc glycopeptide fragments of RNA-polymerase II and mammalian neurofilaments Ernst Meinjohanns Antonio Vargas-Berenguel Morten Meldal Hans Paulsen and Klaus Bock pg 2165; DOI: 10.1039/P19950002165 |
Selective synthesis of unsymmetrical 2,2-dihydroxylated biaryls via electrophilic arylation of metal phenolates with p-benzoquinone monoketals Giovanni Sartori Raimondo Maggi Franca Bigi Simone Giacomelli Cecilia Porta Attilio Arienti and Gabriele Bocelli pg 2177; DOI: 10.1039/P19950002177 |
Facial selectivity in the hydroboration of androst-4-enes James R. Hanson Peter B. Hitchcock Mansur D. Liman and Sivajini Nagaratnam pg 2183; DOI: 10.1039/P19950002183 |
4-Hydroxymethyl steroids related to aphidicolin Juliette A. Boynton and James R. Hanson pg 2189; DOI: 10.1039/P19950002189 |
Synthesis of the glycidol (1R,2R)-1-iodo-2-(triphenylsilyloxy)cyclopropane: new rearrangements of 2,3-epoxy-3-(trialkyl/arylsilyl)-propan-1-ols Barbara Achmatowicz Piotr Raubo and Jerzy Wicha pg 2193; DOI: 10.1039/P19950002193 |
Corrigenda Marcel S. F. Lie Ken Jie Prabhavathi Kalluri Yang Yu Naoto Watanabe Masatomi Ohno and Shoji Eguchi pg 2197; DOI: 10.1039/P19950002197 |
Conference diary pg viim; DOI: 10.1039/P1995000viim |
Front cover pg X073; DOI: 10.1039/P199500FX073 |
Back cover pg X075; DOI: 10.1039/P199500BX075 |
Contents pages pg P195; DOI: 10.1039/P199500FP195 |
Back matter pg P205; DOI: 10.1039/P199500BP205 |
Stereospecific and regiospecific ring opening of glycidol with primary and secondary alcohols mediated by diisobutylaluminium hydride Ravi Kumar Erukulla Hoe-Sup Byun David C. Locke and Robert Bittman pg 2199; DOI: 10.1039/P19950002199 |
Effective, direct biomimetic synthesis of dibenzocyclooctene lignans by hypervalent iodine oxidation of phenolic dibenzylbutyrolactones Andrew Pelter Peter Satchwell Robert S. Ward and Keith Blake pg 2201; DOI: 10.1039/P19950002201 |
Enzymatic esterification and de-esterification of carbohydrates: synthesis of a naturally occurring rhamnopyranoside of p-hydroxybenzaldehyde and a systematic investigation of lipase-catalysed acylation of selected arylpyranosides Nazir B. Bashir Sara J. Phythian Andrew J. Reason and Stanley M. Roberts pg 2203; DOI: 10.1039/P19950002203 |
Enzyme mimics based on cyclic porphyrin oligomers: strategy, design and exploratory synthesis Harry L. Anderson and Jeremy K. M. Sanders pg 2223; DOI: 10.1039/P19950002223 |
Ligand binding by butadiyne-linked porphyrin dimers, trimers and tetramers Harry L. Anderson Sally Anderson and Jeremy K. M. Sanders pg 2231; DOI: 10.1039/P19950002231 |
Template-directed synthesis of linear and cyclic butadiyne-linked porphyrin oligomers up to a linear octamer Sally Anderson Harry L. Anderson and Jeremy K. M. Sanders pg 2247; DOI: 10.1039/P19950002247 |
The roles of templates in the syntheses of porphyrin oligomers Sally Anderson Harry L. Anderson and Jeremy K. M. Sanders pg 2255; DOI: 10.1039/P19950002255 |
A platinum-linked porphyrin trimer and a complementary aluminium tris[3-(4-pyridyl)acetylacetonate] guest Lindsey G. Mackay Harry L. Anderson and Jeremy K. M. Sanders pg 2269; DOI: 10.1039/P19950002269 |
Octatetrayne-linked porphyrins: stretched cyclic dimers and trimers with very spacious cavities Harry L. Anderson Christopher J. Walter Anton Vidal-Ferran Robert A. Hay Philip A. Lowden and Jeremy K. M. Sanders pg 2275; DOI: 10.1039/P19950002275 |
Synthesis of 9-[cis-3-(hydroxymethyl)cyclobutyl]-adenine and -guanine Vijay Kaiwar Colin B. Reese Emily J. Gray and Stephen Neidle pg 2281; DOI: 10.1039/P19950002281 |
Generation of trimethylsulfonium cation from dimethyl sulfoxide and dimethyl sulfate: implications for the synthesis of epoxides from aldehydes and ketones Julie Forrester Ray V. H. Jones Peter N. Preston and Elizabeth S. C. Simpson pg 2289; DOI: 10.1039/P19950002289 |
Heterodiene cycloadditions of C2 symmetric 4,5-disubstituted ketene acetals: the nett asymmetric conjugate addition of recyclable acetic ester enolate equivalents to an activated enone Timothy W. Wallace Ian Wardell Ke-Dong Li Peter Leeming Alan D. Redhouse and S. Richard Challand pg 2293; DOI: 10.1039/P19950002293 |
Amino acids and peptides. Part 42. Application of the 2-adamantyloxycarbonyl (2-Adoc) group to the protection of the imidazole function of histidine in peptide synthesis Yasuhiro Nishiyama Noriyuki Shintomi Yukihiro Kendo Takako Izumi and Yoshio Okada pg 2309; DOI: 10.1039/P19950002309 |
Iron(III) mediated transformations of cyclopropyltrimethylsilyl ethers. Part 1. Free radical tandem ring expansion–cyclisation reactions for the rapid construction of [n.3.0] bicyclic ring systems Kevin I. Booker-Milburn and David F. Thompson pg 2315; DOI: 10.1039/P19950002315 |
Synthesis of 3-alkylpyridines. Part 2. Synthesis of both enantiomers of niphatesine C2 Franz Bracher and Thomas Papke pg 2323; DOI: 10.1039/P19950002323 |
Cyclic peptides from higher plants. Part 21. Thionation of the antitumour cyclic pentapeptides, astins A, B and C, from Aster tataricus Hiroshi Morita Shinji Nagashima Koichi Takeya and Hideji Itokawa pg 2327; DOI: 10.1039/P19950002327 |
Reaction of ortho-lithiated protected anilines with o-hydroxycarbonyl compounds: formation of quino- and pyranoquino-acridines Catherine Jolivet Christian Rivalle Christiane Huel and Emile Bisagni pg 2333; DOI: 10.1039/P19950002333 |
Chiral crown ethers incorporating D-glucose Puthuparampil P. Kanakamma Neelakandha S. Mani Uday Maitra and Vijay Nair pg 2339; DOI: 10.1039/P19950002339 |
Fumiquinazolines A–G, novel metabolites of a fungus separated from a Pseudolabrus marine fish Chika Takahashi Tomochika Matsushita Mitsunobu Doi Katsuhiko Minoura Tetsuro Shingu Yuko Kumeda and Atsushi Numata pg 2345; DOI: 10.1039/P19950002345 |
Total synthesis of balanol: a potent protein kinase C inhibitor of fungal origin C. P. Adams S. M. Fairway C. J. Hardy D. E. Hibbs M. B. Hursthouse A. D. Morley B. W. Sharp N. Vicker and I. Warner pg 2355; DOI: 10.1039/P19950002355 |
Heterocyclic transformations. Part 7. Unprecedented transformations of 1,3-dialkyl-5-formyluracils to 1,3-dialkyl-7-hydroxyquinazolines Harjit Singh Palwinder Singh Swapandeep Singh Chimni and Subodh Kumar pg 2363; DOI: 10.1039/P19950002363 |
Conference diary pg ixb; DOI: 10.1039/P19950000ixb |
Front cover pg X077; DOI: 10.1039/P199500FX077 |
Back cover pg X079; DOI: 10.1039/P199500BX079 |
Contents pages pg P207; DOI: 10.1039/P199500FP207 |
Back matter pg P217; DOI: 10.1039/P199500BP217 |
Acylnitrilium ion initiated spiroannulations in heterocycle synthesis: an application directed toward the total synthesis of the Lycopodium alkaloid ()-serratine Gregory Luedtke and Tom Livinghouse pg 2369; DOI: 10.1039/P19950002369 |
On the scope of acylnitrilium ion initiated heteroannulations: monocyclizations terminated by unactivated alkenes David J. Hughes and Tom Livinghouse pg 2373; DOI: 10.1039/P19950002373 |
Se-Demethylation from 8-dimethylamino-1-methylselanylnaphthalene and its Se-oxide: an X-ray structure of a stable selenenic anhydride with a 8-dimethylamino-1-naphthyl ligand: peri Se N interaction Hisashi Fujihara Hitomi Tanaka and Naomichi Furukawa pg 2375; DOI: 10.1039/P19950002375 |
Unusual behaviour of 4,5-dichloro-1,2,3-dithiazolium chloride (Appel's salt) with 5-aminopyrazoles: a synthetic method of 1H-pyrazolo[3,4-d]thiazoles Gerrit L'abbé Bart D'hooge and Wim Dehaen pg 2379; DOI: 10.1039/P19950002379 |
New synthesis of unsymmetrical dithia compounds Keith Smith and Michael Tzimas pg 2381; DOI: 10.1039/P19950002381 |
Uncatalysed trimethylsilyl cyanide addition to aldehydes Kavita Manju and Sanjay Trehan pg 2383; DOI: 10.1039/P19950002383 |
Pyrylium salts in polyene natural product synthesis: organometallic additions to 4-methylpyrylium tetrafluoroborate Richard J. K. Taylor Karl Hemming and Edna Faria De Medeiros pg 2385; DOI: 10.1039/P19950002385 |
Intramolecular Diels–Alder reactions of the furan diene (IMDAF); rapid construction of highly functionalised isoquinoline skeletons Tomas Hudlicky Gabor Butora Stephen P. Fearnley Andrew G. Gum P. J. Persichini III Michele R. Stabile and Joseph S. Merola pg 2393; DOI: 10.1039/P19950002393 |
Biosynthesis of the dialkylmaleic anhydride-containing antibiotics, tautomycin and tautomycetin Makoto Ubukata Xing-Chun Cheng Jun Uzawa and Kiyoshi Isono pg 2399; DOI: 10.1039/P19950002399 |
Highly asymmetric Pummerer-type cyclization of chiral, non-racemic -amido sulfoxides Yasuyuki Kita Norio Shibata Noriyuki Kawano Takashi Tohjo Chino Fujimori Keita Matsumoto and Shigekazu Fujita pg 2405; DOI: 10.1039/P19950002405 |
Asymmetric aldol reactions of achiral 2-phenylsulfanyl aldehydes with small- and medium-sized carbocyclic rings: the synthesis of homochiral spirocyclic lactones, pyrrolidines and tetrahydrofurans Kelly Chibale and Stuart Warren pg 2411; DOI: 10.1039/P19950002411 |
Reactions of ethyl 2-acetyl-2-azabicyclo[2.2.1]hept-5-ene-3-carboxylate and 4-acetylamino-2-oxabicyclo[3.3.0]oct-7-en-3-one with some electrophiles Michael B. Hursthouse K. M. Abdul Malik David E. Hibbs Stanley M. Roberts Amanda J. H. Seago Vladimir ik and Richard Storer pg 2419; DOI: 10.1039/P19950002419 |
Synthesis and reactivity of iron carbonyl complexes of -silyl substituted ,-unsaturated ketones Susan E. Gibson (née Thomas) and Gary J. Tustin pg 2427; DOI: 10.1039/P19950002427 |
Reactivity of the carbonyl group in water. Generation of azomethine ylides from aqueous formaldehyde: Michael addition versus dipolar trapping André Lubineau Giliane Bouchain and Yves Queneau pg 2433; DOI: 10.1039/P19950002433 |
Ring-opening of N-tosyl aziridines by 2-lithiodithianes William Howson Helen M. I. Osborn and Joseph Sweeney pg 2439; DOI: 10.1039/P19950002439 |
Synthesis and sweet taste of optically active (–)-haematoxylin and of some ()-haematoxylin derivatives Anna Arnoldi Angela Bassoli Gigliola Borgonovo and Lucio Merlini pg 2447; DOI: 10.1039/P19950002447 |
Novel and unexpected one-pot synthesis of 7,7-dioxo-14-oxa-76-thiadibenzo[a,j]anthracene-2,12-disulfonic acid from -tetralone M Fé de la Torre M Luisa Mussons César Raposo José Luis López Josefa Anaya M Cruz Caballero and Joaquín R. Morán pg 2455; DOI: 10.1039/P19950002455 |
Substrate structure and incubation-parameter-dependent selectivities in chiral discrimination of galactopyranosides by -galactosidase hydrolysis Barbara Werschkun Wilfried A. König Vladimír Ken and Joachim Thiem pg 2459; DOI: 10.1039/P19950002459 |
Synthesis of imidazole 1-oxides from 1,2-diimines Jesús Alcázar Mikael Begtrup and Antonio de la Hoz pg 2467; DOI: 10.1039/P19950002467 |
-Substituted pyrrole-based silyl dienol ethers as -amino acid enolate equivalents: a versatile entry to racemic -substituted -amino acids Franca Zanardi Lucia Battistini Gloria Rassu Mara Cornia and Giovanni Casiraghi pg 2471; DOI: 10.1039/P19950002471 |
1,5-Asymmetric induction in reactions between aldehydes and [(4S)-5-(tert-butyldimethylsilyloxy)-4-hydroxypent-2-enyl](tributyl)-stannane promoted by tin(IV) chloride Robert J. Maguire and Eric J. Thomas pg 2477; DOI: 10.1039/P19950002477 |
Stereoselective synthesis of cis- and trans-2,6-disubstituted 5,6-dihydro-2H-pyrans based on 1,5-asymmetric induction in reactions between allylstannanes and aldehydes promoted by tin(IV) chloride Robert J. Maguire and Eric J. Thomas pg 2487; DOI: 10.1039/P19950002487 |
Ag+ Ion-selective lariat ethers: high pressure syntheses and cation recognition properties Kiyoshi Matsumoto Masao Hashimoto Mitsuo Toda and Hiroshi Tsukube pg 2497; DOI: 10.1039/P19950002497 |
Metallation of pyridine N-oxides and application to synthesis Olivier Mongin Patrick Rocca Laurence Thomas-dit-Dumont François Trécourt Francis Marsais Alain Godard and Guy Quéguiner pg 2503; DOI: 10.1039/P19950002503 |
Ozonolysis of (cyclohexa-1,4-dienyl)-L-alanine. An approach to the synthesis of new unnatural amino acids. X-Ray molecular structure of 2-hydroxy-7-methyl-3-phenylpyrazolo[1,5-a]pyrimidine Gury Zvilichovsky and Vadim Gurvich pg 2509; DOI: 10.1039/P19950002509 |
Photoinduced electron-transfer reactions of homonaphthoquinones with amine and arene donors Hiroshi Moriwaki Takumi Oshima and Toshikazu Nagai pg 2517; DOI: 10.1039/P19950002517 |
Conference diary pg ixc; DOI: 10.1039/P19950000ixc |
Front cover pg X081; DOI: 10.1039/P199500FX081 |
Back cover pg X083; DOI: 10.1039/P199500BX083 |
Journals bulletin pg X085; DOI: 10.1039/P1995000X085 |
Contents pages pg P219; DOI: 10.1039/P199500FP219 |
Back matter pg P229; DOI: 10.1039/P199500BP229 |
Use of cyclodextrins to limit product inhibition of (S)-phenylalanine ammonia lyase Christopher J. Easton Jason B. Harper and Stephen F. Lincoln pg 2525; DOI: 10.1039/P19950002525 |
Oxidation of some prochiral 3-substituted cyclobutanones using monooxygenase enzymes: a single-step method for the synthesis of optically enriched 3-substituted -lactones René Gagnon Gideon Grogan Esther Groussain Sandrine Pedragosa-Moreau Paul F. Richardson Stanley M. Roberts Andrew J. Willetts Véronique Alphand Jacques Lebreton and Roland Furstoss pg 2527; DOI: 10.1039/P19950002527 |
Short synthetic approach towards the triindenotriphenylene (hemifullerene) system G. Mehta G. V. Raghava Sharma (the late) M. A. Krishna Kumar T. V. Vedavyasa and E. D. Jemmis pg 2529; DOI: 10.1039/P19950002529 |
Aryllead-mediated synthesis of linear 3-arylpyranocoumarins: synthesis of robustin and robustic acid Dervilla M. X. Donnelly David J. Molloy John P. Reilly and Jean-Pierre Finet pg 2531; DOI: 10.1039/P19950002531 |
Regio- and enantio-selective enolisations of cyclic ketones using chiral lithium amide bases Kimberley Bambridge Barry P. Clark and Nigel S. Simpkins pg 2535; DOI: 10.1039/P19950002535 |
Synthesis, X-ray structure, thermal stability and reactions of triaryl(3-oxoalkyl)bismuthonium salts Yoshihiro Matano Nagao Azuma and Hitomi Suzuki pg 2543; DOI: 10.1039/P19950002543 |
Steric acceleration of intramolecular oxime and hydrazone cycloadditions Jane E. Bishop Katherine A. Flaxman Barry S. Orlek Peter G. Sammes and David J. Weller pg 2551; DOI: 10.1039/P19950002551 |
Bis(hydroxyphenyloxazolinato)-titanium(IV) and -zirconium(IV) triflates as novel transition metal-based Lewis acids Pier Giorgio Cozzi and Carlo Floriani pg 2557; DOI: 10.1039/P19950002557 |
Benzazepine formation by the 1.7 electrocyclisations of diene-conjugated nitrile ylides: studies on relative rates of cyclisation via intramolecular competition reactions Kevin E. Cullen and John T. Sharp pg 2565; DOI: 10.1039/P19950002565 |
Synthesis of 17H-tetrabenzo[a,c,g,i]fluorene derivatives as chiral selectors for enantiomeric separation by HPLC on porous graphitised carbon Jonathan K. Dutton John H. Knox Xavier Radisson Harold J. Ritchie and Robert Ramage pg 2581; DOI: 10.1039/P19950002581 |
Synthesis of photoresponsive crown ethers having a phosphoric acid functional group as anionic cap and their selective complexing abilities toward alkali metal cations Sadatoshi Akabori Yoshikazu Miura Noriko Yotsumoto Kiyoshi Uchida Masaru Kitano and Yoichi Habata pg 2589; DOI: 10.1039/P19950002589 |
Synthesis of some -trichloromethyl-azines and -diazines David Cartwright John R. Ferguson Thomas Giannopoulos George Varvounis and Basil J. Wakefield pg 2595; DOI: 10.1039/P19950002595 |
Asymmetric formal total synthesis of (–)-swainsonine Wei-Shan Zhou Wen-Ge Xie Zhi-Hui Lu and Xin-Fu Pan pg 2599; DOI: 10.1039/P19950002599 |
Reaction of N-arylsulfonylaziridines with dimethylsulfoniumethoxycarbonyl methylide: regio- and stereo-selective synthesis of 1-arylsulfonyl-2-ethoxycarbonyl azetidines Upender K. Nadir and Anjali Arora pg 2605; DOI: 10.1039/P19950002605 |
Novel synthesis of 5,10,15,20-tetraarylporphyrins using high-valent transition metal salts Ana Gradillas Carmen del Campo José V. Sinisterra and Emilio F. Llama pg 2611; DOI: 10.1039/P19950002611 |
Atropisomer-selective ligand-coupling reactions of sulfoxides. X-Ray molecular and crystal structures for 2-({2-(4-chlorophenyl)naphtho[1,2-b]thiophen-3-yl}amino)-2-methylpropan-1-ol, 2-(2-hydroxy-1,1-dimethylethyl)-2,3-dihydronaphtho[2,1-d]isothiazol-3-one and (R)-(+)-2-bromo-1-(tert-butylsulfinyl)naphthalene Robert W. Baker David C. R. Hockless Geoffrey R. Pocock Melvyn V. Sargent Brian W. Skelton Alexander N. Sobolev Edi Twiss (née Stanojevic) and Allan H. White pg 2615; DOI: 10.1039/P19950002615 |
Lewis acid induced N-methyleneamine equivalents. Part 3. Addition of allyl nucleophiles to TiCl4-induced N-methyleneamine equivalents: synthesis of 1,2,3,4-tetrahydroquinolines and homoallylic anilines Hyun-Joon Ha Young-Gil Ahn and Jung-Kyoon Chon pg 2631; DOI: 10.1039/P19950002631 |
Photocycloaddition-cyclobutane rearrangement to spiro cyclopentanones: application in a formal synthesis of ()--cedrene Debasis Patra and Subrata Ghosh pg 2635; DOI: 10.1039/P19950002635 |
2-Azaallyl anions: key models for the elaboration of alkyl-, amino- and hydroxy-1,7-naphthyridine derivatives Axel Couture Pierre Grandclaudon Cristian Simion and Patrice Woisel pg 2643; DOI: 10.1039/P19950002643 |
Synthetic application of biotransformations: absolute stereochemistry and Diels–Alder reactions of the (1S,2R)-1,2-dihydroxycyclohexa-3,5-diene-1-carboxylic acid from Pseudomonas putida Gareth N. Jenkins Douglas W. Ribbons David A. Widdowson Alexandra M. Z. Slawin and David J. Williams pg 2647; DOI: 10.1039/P19950002647 |
ipso-vs. tele-Nucleophilic substitution by piperidine on isocolchicides and colchicides bearing an -leaving group Marino Cavazza and Francesco Pietra pg 2657; DOI: 10.1039/P19950002657 |
Synthesis and cycloaddition of 2,4-dihydropyrrolo[3,4-b]indoles Arumugasamy Jeevanandam and Panayencheri C. Srinivasan pg 2663; DOI: 10.1039/P19950002663 |
Conference diary pg ixd; DOI: 10.1039/P19950000ixd |
Front cover pg X089; DOI: 10.1039/P199500FX089 |
Back cover pg X091; DOI: 10.1039/P199500BX091 |
Contents pages pg P231; DOI: 10.1039/P199500FP231 |
Stereoselective synthesis of 3--D-ribofuranosylpyrazole from 2,3-O-isopropylidene-D-ribose; a new route to pyrazole C-nucleosides Anthony D. Rycroft Gurdial Singh and Richard H. Wightman pg 2667; DOI: 10.1039/P19950002667 |
Samarium diiodide promoted coupling of thiophenecarbaldehydes Shyh-Ming Yang and Jim-Min Fang pg 2669; DOI: 10.1039/P19950002669 |
Enantioselective synthesis of -arylpropanoic acids Philip C. Bulman Page Michael J. McKenzie and Derek R. Buckle pg 2673; DOI: 10.1039/P19950002673 |
Facile synthesis of the key intermediate of EO 9 via the formation of the indole skeleton using the Nenitzescu reaction Masahiko Kinugawa Hitoshi Arai Hiroshi Nishikawa Akihiko Sakaguchi Takehiro Ogasa Shinji Tomioka and Masaji Kasai pg 2677; DOI: 10.1039/P19950002677 |
Facile retro-cycloaddition of adducts derived from steroidal 5,7-diene and 4-phenyl-1,2,4-triazoline-3,5-dione by diisobutylaluminium hydride Fumihiro Kondo Misako Miyashita Katsuhiro Konno and Hiroaki Takayama pg 2679; DOI: 10.1039/P19950002679 |
Preparation and direct observation by 19F NMR spectroscopy of 1-fluoro-1-lithioalkenes Andrew Pelter Jaroslav Kvicala and David E. Parry pg 2681; DOI: 10.1039/P19950002681 |
Novel synthesis of 3-chloromethylidene-2-ethoxy-1,25-oxaphospholan-2-ones catalysed by palladium(II) Chunlin Ma Xiyan Lu and Yongxiang Ma pg 2683; DOI: 10.1039/P19950002683 |
Active conformation of the inositol monophosphatase substrate, adenosine 2-phosphate: role of the ribofuranosyl O-atoms in chelating a second Mg2+ ion Andrew G. Cole and David Gani pg 2685; DOI: 10.1039/P19950002685 |
Probes for the position and mechanistic role of the second catalytic magnesium ion in the inositol monophosphatase reaction Andrew G. Cole John Wilkie and David Gani pg 2695; DOI: 10.1039/P19950002695 |
3-Dimensional interactions between inositol monophosphatase and its substrates, inhibitors and metal ion cofactors John Wilkie Andrew G. Cole and David Gani pg 2709; DOI: 10.1039/P19950002709 |
The lithiation of fluorinated benzenes and its dependence on solvent and temperature Paul Leslie Coe Anthony John Waring and Thomas David Yarwood pg 2729; DOI: 10.1039/P19950002729 |
Synthesis of 4-phenylpiperidines by tandem Wittig olefination–aza-Wittig rearrangement of 2-benzoylaziridines Iain Coldham Alan J. Collis Roger J. Mould and Richard E. Rathmell pg 2739; DOI: 10.1039/P19950002739 |
Synthesis of ()-aklavinone and ()-auramycinone via electron-deficient o-quinonoid pyrones David W. Jones and Christopher J. Lock pg 2747; DOI: 10.1039/P19950002747 |
LICKOR-Promoted 1,2-elimination in 1,1-dimethoxy-2-phenylethane and 1,1-dimethoxy-2-phenylpropane: synthesis of substituted enol ethers and alkynes Annamaria Deagostino Mariella Mella Cristina Prandi and Paolo Venturello pg 2757; DOI: 10.1039/P19950002757 |
Regio- and stereo-selective synthesis of trifluoromethylated isoxazolidines by 1,3-dipolar cycloaddition of 1,1,1-trifluoro-3-phenylsulfonylpropene with nitrones, and their conversion into trifluoromethylated syn-3-amino alcohols Hiroyasu Tsuge Takashi Okano and Shoji Eguchi pg 2761; DOI: 10.1039/P19950002761 |
Synthesis of some analogues of cytisine: unusual reduction pathways for tertiary nitro groups in sterically constrained molecules Kristina J. Blackall David Hendry Robert J. Pryce and Stanley M. Roberts pg 2767; DOI: 10.1039/P19950002767 |
Synthesis of 4-hydroxylamino-1-azabuta-1,3-dienes and their cyclization to 2-substituted pyrazole 1-oxides Jesús Alcazar Inés Almena Mikael Begtrup and Antonio de la Hoz pg 2773; DOI: 10.1039/P19950002773 |
Antitumour imidazotetrazines. Part 33. New syntheses of the antitumour drug temozolomide using masked methyl isocyanates Yongfeng Wang Malcolm F. G. Stevens William T. Thomson and Bruce P. Shutts pg 2783; DOI: 10.1039/P19950002783 |
Ligand coupling and neighbouring-group effects in the alkaline hydrolysis of arylphosphonium salts: new stable tetraarylphosphonium benzimidazolate betaines David W. Allen and Peter Benke pg 2789; DOI: 10.1039/P19950002789 |
Synthesis of 1,6-diethynylcyclohepta-1,3,5-triene and its oxidative coupling to dimethano-bridged octadehydro[20]annulene and trimethano-bridged dodecadehydro[30]annulene Jro Ojima Tomoyo Daimon Naoki Hiraiwa Hiroyuki Higuchi Masako Ueno and Gaku Yamamoto pg 2795; DOI: 10.1039/P19950002795 |
Diastereoselectivity and assignment of absolute stereochemistry in the aza-Diels–Alder reaction of a sulfonylimino acetate with 1-methoxy-3-trimethylsilyloxybuta-1,3-diene Andrew K. McFarlane Gareth Thomas and Andrew Whiting pg 2803; DOI: 10.1039/P19950002803 |
Corrigendum A. V. Nikolaev T. J. Rutherford M. A. J. Ferguson and J. S. Brimacombe pg 2809; DOI: 10.1039/P19950002809 |
Conference diary pg ixe; DOI: 10.1039/P19950000ixe |
Front cover pg X093; DOI: 10.1039/P199500FX093 |
Back cover pg X095; DOI: 10.1039/P199500BX095 |
Contents pages pg P241; DOI: 10.1039/P199500FP241 |
Assembly of bicyclo[2.2.1]heptane derivatives by two types of domino reaction Masataka Ihara Shuichi Suzuki Yuji Tokunaga and Keiichiro Fukumoto pg 2811; DOI: 10.1039/P19950002811 |
Cyclopenta[a]phenalen-9(8H)-one: an extended phenalenone system Yoshikazu Sugihara Reiko Hashimoto Hitoshi Fujita Noritaka Abe Hiromasa Yamamoto Takashi Sugimura and Ichiro Murata pg 2813; DOI: 10.1039/P19950002813 |
Characterization of an imidazolium compound formed by reaction of methylglyoxal and N-hippuryllysine Elisabeth Brinkmann Kevin J. Wells-Knecht Suzanne R. Thorpe and John W. Baynes pg 2817; DOI: 10.1039/P19950002817 |
Studies in the cycloproparene series; heterocyclic substituted methylidenecyclopropa[b]naphthalenes Brian Halton Mark J. Cooney Tim W. Davey Grant S. Forman Qi Lu Roland Boese Dieter Bläser and Andreas H. Maulitz pg 2819; DOI: 10.1039/P19950002819 |
Mechanistic studies of a Pummerer-type reaction in acyclic and rigid cyclic sulfoxides induced by ketene tert-butyldimethylsilyl methyl acetal Yasuyuki Kita Norio Shibata Naoki Yoshida Noriyuki Kawano Chino Fujimori Naoki Yoshikawa and Shigekazu Fujita pg 2829; DOI: 10.1039/P19950002829 |
New route to 1-formylalkylphosphonates using diethyl trichloromethylphosphonate as a precursor Yannick Zanella Sylvie Berté-Verrando Rachel Dizière and Philippe Savignac pg 2835; DOI: 10.1039/P19950002835 |
Stereochemical and mechanistic studies on the formation of the 3-oxoindolizidine skeleton from ornithine derivatives M José Domínguez M Teresa García-López Rosario Herranz Mercedes Martín-Martínez and Rosario González-Muñiz pg 2839; DOI: 10.1039/P19950002839 |
Rearrangement of 1-phenyl-3,4-dihydro-1H-2-benzothiopyranium 2-methylides Toru Tanzawa Naohiro Shirai Yoshiro Sato Keiichiro Hatano and Yukihisa Kurono pg 2845; DOI: 10.1039/P19950002845 |
Highly stereocontrolled total synthesis of (+)-bengamide E Chisato Mukai Sameh M. Moharram Osamu Kataoka and Miyoji Hanaoka pg 2849; DOI: 10.1039/P19950002849 |
Synthesis of arizonin C1 Margaret A. Brimble Sara J. Phythian and Hishani Prabaharan pg 2855; DOI: 10.1039/P19950002855 |
Syntheses of 6-hydroxyshikimic acid and its derivatives A. John Blacker R. John Booth Gareth M. Davies and James K. Sutherland pg 2861; DOI: 10.1039/P19950002861 |
Synthesis of chiral diferrocenyl dichalcogenides and their application to asymmetric nucleophilic ring opening of meso-epoxides Yoshiaki Nishibayashi Jai Deo Singh Shin-ichi Fukuzawa and Sakae Uemura pg 2871; DOI: 10.1039/P19950002871 |
(2R, 3S)- and (2S, 3R)-2-Benzyl-3,4-epoxybutanoic acid as highly efficient and fast acting pseudomechanism-based inactivators for carboxypeptidase a: design, asymmetric synthesis and inhibitory kinetics Soo Suk Lee Zhi-Hong Li Dong Ha Lee and Dong H. Kim pg 2877; DOI: 10.1039/P19950002877 |
Synthesis of aliphatic O-dimannosyl amino acid building blocks for solid-phase assembly of glycopeptide libraries Henrik Franzyk Morten Meldal Hans Paulsen and Klaus Bock pg 2883; DOI: 10.1039/P19950002883 |
Activity and enantioselectivity of serine proteases in transesterification reactions in organic media Jaap Broos Johan F. J. Engbersen Inna K. Sakodinskaya Willem Verboom and David N. Reinhoudt pg 2899; DOI: 10.1039/P19950002899 |
Heterocyclizations of 3-trifluoroacetyl substituted lactams with cyclic 1,3-bis-nucleophiles Jean-Philippe Bouillon Zdenek Janousek Heinz G. Viehe Bernard Tinant and Jean-Paul Declercq pg 2907; DOI: 10.1039/P19950002907 |
Diastereoselective allylation of chiral sulfinyl-substituted thiophenecarbaldehydes with a Lewis acid Yoshitsugu Arai Atsuko Suzuki Tsutomu Masuda Yukio Masaki and Motoo Shiro pg 2913; DOI: 10.1039/P19950002913 |
trans-Fused crown ethers from 2,5-O-methylene-D-mannitol: synthesis, X-ray diffraction structure and full nuclear magnetic resonance spectroscopic data of 1,6-diazido-1,6-dideoxy-2,5-O-methylene-3,4-O-naphthalene-2,3-diylbis(oxyethyleneoxyethylene)-D-mannitol and 3,4-di-O-acetyl-1,6-diazido-1,6-dideoxy-2,5-O-methylene-D-mannitol Mostafa Nazhaoui Jean-Pierre A. Joly Bertrand J. Jean-Claude Valerio Del Duca André Aubry and Mohammed Boubouh pg 2919; DOI: 10.1039/P19950002919 |
(Z)-Heptadec-8-enylboronic acid: a potential lipase inhibitor Valeri Martichonok and J. Bryan Jones pg 2927; DOI: 10.1039/P19950002927 |
Photochemistry of the nitrogen–thiocarbonyl systems. Part. 24. Photoreactions of thiobenzamide with various substituted furans: regioselective -benzoylation and transformation of furans to other aromatic compounds Kazuaki Oda Hisao Tsujita Kosei Ohno and Minoru Machida pg 2931; DOI: 10.1039/P19950002931 |
Diacetylenic sterols: new potentially photopolymerizable lipids Catherine Vilchèze and Robert Bittman pg 2937; DOI: 10.1039/P19950002937 |
Preparation of thiazolocarbazoles via the Fischer indole synthesis Laurent Martarello Delphine Joseph and Gilbert Kirsch pg 2941; DOI: 10.1039/P19950002941 |
Reactivity of cyclic arsenites and phosphites: X-ray structures of bis(5,5-dimethyl-1,3,2-dioxarsenan-2-yl) ether and bis(2,4,8,10-tetra-tert-butyl-12H-dibenzo [d,g][1,3,2]dioxarsenocin-6-yl) ether Musa A. Said K. C. Kumara Swamy M. Veith and V. Huch pg 2945; DOI: 10.1039/P19950002945 |
Conference diary pg ixf; DOI: 10.1039/P19950000ixf |
Front cover pg X097; DOI: 10.1039/P199500FX097 |
Back cover pg X099; DOI: 10.1039/P199500BX099 |
Contents pages pg P251; DOI: 10.1039/P199500FP251 |
Back matter pg P259; DOI: 10.1039/P199500BP259 |
Alkoxycarbonyl groups transfer to amines by the N,N-dibenzyl-and N,N-di-tert-butyl-carbamates of cyclic thioureas Noboru Matsumura Akiko Noguchi Aya Kitayoshi and Hiroo Inoue pg 2953; DOI: 10.1039/P19950002953 |
Facile and stereospecific synthesis of 1,1-dihalogenoalk-1-enes from 1-halogenoalk-1-ynes by hydroboration Yuzuru Masuda Toshihiro Suyama Miki Murata and Shinji Watanabe pg 2955; DOI: 10.1039/P19950002955 |
Novel stereoselective incorporation and hydrolysis of long-chain amino-acid substrates by vesicular membrane systems which include tri- or tetra-peptide catalysts Katsutoshi Ohkubo Kenji Urabe Junji Yamamoto Takashi Sagawa and Satoshi Usui pg 2957; DOI: 10.1039/P19950002957 |
Kinetic resolution of alcohols in an asymmetric mitsunobu reaction using chiral nonracemic 1,3,2-dioxaphosphepanes Ron Hulst Arjan van Basten Kevin Fitzpatrick and Richard M. Kellogg pg 2961; DOI: 10.1039/P19950002961 |
Regiospecific synthesis of 4-fluoro-4,3-keto steroids using caesium fluoroxysulfate Harold F. Hodson David J. Madge and David A. Widdowson pg 2965; DOI: 10.1039/P19950002965 |
Biotransformation of -unsaturated carbonyl compounds: sulfides, sulfoxides, sulfones, nitriles and esters by yeast species: carbonyl group and carbon–carbon double bond reduction Surinder Koul David H. G. Crout William Errington and Jiri Tax pg 2969; DOI: 10.1039/P19950002969 |
New entry to a cis-fused bicyclic ring system by a [2,3]sigmatropic rearrangement via cyclic allylsulfonium ylides. Synthesis of the cis-2-oxa-9-vinyldecalin skeleton Fusao Kido Toshiya Abiko and Michiharu Kato pg 2989; DOI: 10.1039/P19950002989 |
Highly regioselective access to 7-substituted 1,4,7,10-tetraazacyclododecane-1-carbaldehyde derivatives: synthetic aspects and NMR elucidation of the structures. X-Ray crystal structures of 7-triphenylmethyl-1,4,7,10-tetraazacyclododecane-1-carbaldehyde and 7-triphenylmethyloctahydro-5H,9bH-2a,4a,7,9a-tetraazacycloocta [cd] pentalene Pier Lucio Anelli Luisella Calabi Paolo Dapporto Marcella Murru Lino Paleari Paola Paoli Fulvio Uggeri Sandra Verona and Mario Virtuani pg 2995; DOI: 10.1039/P19950002995 |
Oligomeric flavanoids. Part 19. Reductive cleavage of the interflavanyl bond in proanthocyanidins Petrus J. Steynberg Jan P. Steynberg Barend C. B. Bezuidenhoudt and Daneel Ferreira pg 3005; DOI: 10.1039/P19950003005 |
New, short synthesis of arylnaphthofuranone lignans based on reactions of o-aroylbenzyllithiums with furan-2(5H)-one Kazuhiro Kobayashi Junsuke Tokimatsu Kouji Maeda Osamu Morikawa and Hisatoshi Konishi pg 3013; DOI: 10.1039/P19950003013 |
Solid-phase synthesis of a fucosylated glycopeptide of human factor IX with a fucose--(1O)-serine linkage Stefan Peters Todd L. Lowary Ole Hindsgaul Morten Meldal and Klaus Bock pg 3017; DOI: 10.1039/P19950003017 |
Simple and efficient strategy for making -(16)-linked galactooligosaccharides using naked galactopyranosides as acceptors Ravindranathan K. P. Kartha Makoto Kiso Akira Hasegawa and Harold J. Jennings pg 3023; DOI: 10.1039/P19950003023 |
Synthesis and properties of dimethano-bridged tetradehydro[21]-, -[23]- and -[25]annulenones Jro Ojima Naoki Hiraiwa Shiro Kondo Kaori Asano Chiaki Sakon Hiroyuki Higuchi Katsuya Inoue and Gaku Yamamoto pg 3027; DOI: 10.1039/P19950003027 |
Biomimetic iron porphyrin-catalysed oxidation of cyclopenta [a] phenanthrenones Grahame J. Harden and Maurice M. Coombs pg 3037; DOI: 10.1039/P19950003037 |
Synthesis and reactions of 5-benzylidene-2-phenyl-4,5-dihydro-1,3-oxazol-4-ones Yennu Santosh Laxmi and Divi Sarangapani Iyengar pg 3043; DOI: 10.1039/P19950003043 |
Corrigendum Vijay Nair and Jessy Mathew pg 3047; DOI: 10.1039/P19950003047 |
Conference diary pg viin; DOI: 10.1039/P1995000viin |
Front cover pg X101; DOI: 10.1039/P199500FX101 |
Back cover pg X103; DOI: 10.1039/P199500BX103 |
Contents pages pg P261; DOI: 10.1039/P199500FP261 |
Unimolecular chain transfer (UMCT) reactions: concepts, preliminary results with silicon hydrides, and future potential Dennis P. Curran Jinyou Xu and Edoardo Lazzarini pg 3049; DOI: 10.1039/P19950003049 |
Giese-type radical addition reactions to an acceptor that functions by a unimolecular chain transfer reaction of a silicon hydride Dennis P. Curran and Jinyou Xu pg 3061; DOI: 10.1039/P19950003061 |
Design of new phosphonium salt host compounds Fumio Toda Koichi Tanaka and Hirotoshi Sawada pg 3065; DOI: 10.1039/P19950003065 |
Studies on the stereoselectivity of osmylation of cis-bicyclo [3.3.0]-oct-6-enes Nigel Broom Peter J. O'Hanlon Thomas J. Simpson Rosamund Stephen and Christine L. Willis pg 3067; DOI: 10.1039/P19950003067 |
Synthesis of enterochelin Henry J. Rogers pg 3073; DOI: 10.1039/P19950003073 |
Aminolysis and alkaline hydrolysis of protected 1-hydroxybenzo-triazol-1-yl esters of adenosine 5-phosphorothioate and -phosphorodithioate Colin B. Reese Louise H. K. Shek and Zhengyun Zhao pg 3077; DOI: 10.1039/P19950003077 |
Synthesis of cyclocholate-capped porphyrins Richard P. Bonar-Law and Jeremy K. M. Sanders pg 3085; DOI: 10.1039/P19950003085 |
Photochemical reaction of 1-(o-methylaryl)-2,2-dimethyl 1,3-diketones in the presence of oxygen Michikazu Yoshioka Kaori Nishizawa Johji Suzuki Yasuhiro Iwata Shigekazu Kumakura and Tadashi Hasegawa pg 3097; DOI: 10.1039/P19950003097 |
Three positional isomers of substituted triphenylmethanes from reactions of trityl anion with 1-acyl-2,2-dimethylaziridines Jürgen Werry Pen-Yuan Lin Petros Assithianakis and Helmut Stamm pg 3103; DOI: 10.1039/P19950003103 |
Sesqui- and di-terpene biosynthesis from 13C labelled acetate and mevalonate in cultured cells of Heteroscyphus planus Kensuke Nabeta Takehiro Ishikawa and Hiroshi Okuyama pg 3111; DOI: 10.1039/P19950003111 |
Synthesis and oxidative behaviour of reduced indeno[1,2-b]quinoxalines and benzo[b]phenazines David W. Brown Mary F. Mahon Aleyamma Ninan and Malcolm Sainsbury pg 3117; DOI: 10.1039/P19950003117 |
New route to amino[2H2]methylphosphonic acid via bis(trifluoroethyl) phosphonate transesterification Sylvie Berté-Verrando Rachel Dizière Mohammad Samadi and Philippe Savignac pg 3125; DOI: 10.1039/P19950003125 |
Conversions of 2-aminopyridines into 5-substituted derivatives mediated by 1-hydroxymethylbenzotriazole Alan R. Katritzky Saad El-Zemity and Hengyuan Lang pg 3129; DOI: 10.1039/P19950003129 |
Synthesis of the Calophyllum coumarins. Part 2 Christopher J. Palmer and Jonathan L. Josephs pg 3135; DOI: 10.1039/P19950003135 |
Conference diary pg viio; DOI: 10.1039/P1995000viio |